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1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperazine
5-(2H-1,3-benzodioxol-4-ylmethyl)-1-(2-hydroxyethyl)-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
4-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[2-(dimethylamino)ethyl]-8-(5-methoxypyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[4-(methylsulfanyl)phenyl]methyl}piperazine
N-(1-{4-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
N-cyclopropyl-1-(isoquinoline-5-carbonyl)piperazine-2-carboxamide
2-{4-[4-(hydroxymethyl)pyridin-2-yl]phenyl}-2-methylpropanenitrile
(2E)-3-(pyridin-2-yl)-1-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]prop-2-en-1-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(1,2-oxazolidin-2-yl)propanamide
4-[4-(4-methoxyphenyl)-3-oxopiperazine-1-carbonyl]oxane-4-carbonitrile
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
2-[2,4-dioxo-1-(2-phenylethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
N,2-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
N-(furan-2-ylmethyl)-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[2-(2-fluorophenyl)benzoyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-(3-phenylpropyl)pyridin-2-amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-{4-[(2-ethylpyrimidin-4-yl)methyl]-1,4-diazepan-1-yl}-1,3-benzothiazole
2-ethyl-8-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(2-methylphenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxylic acid
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(3-methoxyphenyl)ethan-1-one
1-(pyridin-4-yl)-4-(quinoxaline-6-carbonyl)-1,4-diazepan-6-ol
N-[(3,5-dimethoxyphenyl)methyl]-5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
5-(4-methylpyrimidin-2-yl)thiophene-2-carboxylic acid
(5S)-5-{4-[2-(3-methoxyphenyl)-1-[methyl(pyridin-2-ylmethyl)amino]ethyl]piperidine-1-carbonyl}pyrrolidin-2-one
3-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}benzonitrile
2-(4-acetylphenoxy)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
2-methyl-1-[4-({[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)piperidin-1-yl]propan-1-one
3-[2-(dimethylamino)ethyl]-5-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
4-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-N-methyl-1,3-thiazol-2-amine
{1-[4-(4-chlorophenoxy)piperidin-1-yl]-3-methyl-1-oxobutan-2-yl}urea
N3-cyclooctyl-N5-[(5-fluoro-2-methylphenyl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{[8-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethylfuran-3-carboxamide
3-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-2-methyl-4-phenylpyridine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(pyridin-4-ylmethyl)oxolane-2-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
4-[3-(1H-imidazol-2-yl)piperidin-1-yl]-N,N-dimethyl-5,6,7,8-tetrahydroquinazolin-2-amine
3-{[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}-N-(1,3-thiazol-2-yl)propanamide
2-(4-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
5,8-dimethyl-2-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)quinolin-4-ol
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
methyl 2-(3-methylphenyl)-2-[2-(pyridin-4-yl)acetamido]acetate
N-(2,4-dimethoxyphenyl)-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}propanamide
1-hydroxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]cyclopentane-1-carboxamide
1-(morpholin-4-yl)-3-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]propan-1-one
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine