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N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
methyl({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)[1-(pyridin-4-yl)ethyl]amine
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methylphenyl)methyl]acetamide
methyl 3-(4-chlorobenzoyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[1-(2-methyl-1-benzofuran-5-carbonyl)pyrrolidin-2-yl]pyridine
ethyl 2-{N-methyl-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamido}acetate
N,N-dimethyl-2-{[3-(pyridin-4-yl)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-cyclopropyl-N-[(1S)-1-(4-fluorophenyl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-(cyclopropylmethyl)-3-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
2-[(5-methylpyrazin-2-yl)methyl]-8-(4,4,4-trifluorobutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-1-phenylcyclohexane-1-carboxamide
(1R,5S)-3-(5-ethylpyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-hydroxy-2-methylpropan-2-yl)-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
1-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-2-methylpiperidine
1-cyclopentyl-5-[4-(2-methylphenyl)piperazine-1-carbonyl]piperidin-2-one
N2-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]pyrimidine-2,4-diamine
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)acetamide
1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-4-oxo-N-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
N-ethyl-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(oxolan-2-ylmethyl)benzamide
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(3-methoxyphenyl)methyl]piperidin-3-yl]propanoate
methyl (2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-[(pyrimidin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
1-[2-(2-butoxy-5-methylphenyl)pyridine-4-carbonyl]-4-methylpiperazine
4-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}-N-(pyridin-3-yl)benzamide
5-phenyl-N-(4-{4-[(2,2,2-trifluoroethyl)amino]piperidin-1-yl}phenyl)pentanamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)cyclohexanecarboxamide
methyl 2-[(3,4-difluorophenyl)sulfamoyl]-6-[(2E)-4-methylpent-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-(quinolin-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
6-methyl-2-[(2S)-1-methylpyrrolidine-2-carbonyl]-5-[5-(oxolan-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)propanamide
[1-(pyrimidin-2-yl)piperidin-4-yl](thiophen-2-yl)methanol
7-(3-chlorophenyl)-4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[7-(2-chlorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
2-[3-(2H-1,3-benzodioxol-5-yl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[(1-ethyl-1H-imidazol-2-yl)methyl]benzamide
[(3-chloropyridin-4-yl)methyl]({imidazo[1,2-a]pyridin-3-ylmethyl})methylamine
N-methyl-5-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-[(2-fluorophenyl)methyl]-4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1,4-diazepane
4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1-(3-methoxyphenyl)-5-methylpiperazin-2-one
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
4-[(2S)-2-amino-2-cyclopropylacetyl]-1-(2-phenylphenyl)piperazin-2-one
2-methyl-8-[(4-phenoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine
methyl 7-oxo-3-(2-phenoxypropanoyl)-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]amine
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-4-(thiophen-2-yl)butanamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-tert-butyl-6-[(thiophen-2-ylmethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide