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(3S,4S)-4-(naphthalen-2-yl)-1-(1,3-oxazole-5-carbonyl)piperidin-3-ol
1-(1H-indole-3-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
4-{5-[(2S)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
N-[(3S,4R)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
1-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
methyl 4-{4-[2-(4-hydroxyphenyl)acetyl]piperazin-1-yl}benzoate
3-fluoro-5-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carbonyl}benzonitrile
1-[2-({[(8-chloro-4-hydroxyquinolin-2-yl)methyl]amino}methyl)morpholin-4-yl]ethan-1-one
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
1-({3-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)-3-methoxypyrrolidine
4-(2-methyl-1-benzofuran-5-carbonyl)-1,4-oxazepan-6-ol
4-(4-chlorophenyl)-1-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}butan-1-one
N-methyl-1-(naphthalen-1-ylmethyl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-{3-[4-(2-chlorophenoxy)piperidin-1-yl]-3-oxopropyl}-5-[(4-fluorophenyl)methyl]pyrrolidin-2-one
[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]propanamide
(2R)-2-amino-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-methylpentan-1-one
1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-(1,3-oxazole-5-carbonyl)-1,4-diazepan-6-ol
6-[(3-chlorophenyl)methyl]-N-(3-fluorophenyl)-6-azaspiro[2.5]octane-1-carboxamide
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanoic acid
5-[(4-methylpiperazin-1-yl)methyl]-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)furan-2-carboxamide
(3S,4R)-1-(4-cyanobenzoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
4-[(8-methoxyquinolin-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
({4-ethyl-5-[1-(quinolin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-(1-{[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-[3-(furan-2-yl)-3-phenylpropyl]-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-phenylpropanamide
4-({1-[(2-methylphenyl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
1-[6-(3-methoxyphenoxy)pyridin-3-yl]-3-{2-[(2S)-pyrrolidin-2-yl]ethyl}urea
N-[2-(diethylamino)ethyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]phenyl}pyrrolidin-2-one
4-[2-(2-chloro-6-fluorophenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
N-methyl-N-(1-methylpiperidin-4-yl)-3-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)propanamide
3-({1-[(4-methoxypyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
(3R,4S)-4-{4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-1,4-diazepan-1-yl}oxolan-3-ol
2-[4-({3-[2-(hydroxymethyl)piperidin-1-yl]propyl}amino)-6-methylpyrimidin-2-yl]phenol
4-(3-chloro-4-methoxyphenyl)-3-[1-(propan-2-yloxy)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(methoxymethyl)-N-(3-methyl-1-{7-[(6-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylfuran-3-carboxamide
N-[2-(N-methylmethanesulfonamido)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
methyl 5-[4-(4-methoxybenzoyl)piperazin-1-yl]-5-oxopentanoate
N-{1-[1-(1-carbamoylethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-[(2R,3R)-1'-[(3,5-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
N,2-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-benzothiazole-6-carboxamide
5-methyl-6-({4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}sulfonyl)-2,3-dihydro-1,3-benzoxazol-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-7-(2-methoxyacetamido)-N-methyl-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
3-cyclobutyl-4-(2-ethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-[2-(propan-2-yloxy)ethyl]acetamide
methyl 4-[(butan-2-yl)(pyridin-4-ylmethyl)carbamoyl]benzoate