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2-[1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-[1-(7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclopropanecarboxamide
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2-fluoro-5-methoxyphenyl)methyl]piperidine
2-{3-[1-(dimethylamino)ethyl]phenyl}pyridine-4-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methylnaphthalene-1-carboxamide
N-[(3R,4S)-1-(cyclopropanesulfonyl)-4-cyclopropylpyrrolidin-3-yl]-6-(methoxymethyl)pyrimidin-4-amine
4-(2,3-dihydro-1H-inden-2-yl)-7-(3,6-dimethylpyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(2,6-dimethylphenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
2-{[4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazol-1-yl]methyl}-3,4-dihydroquinazolin-4-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(1-methyl-5-phenyl-1H-pyrazol-3-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[(2-fluorophenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
(2R,3R)-3-amino-1'-(3-propyl-1H-pyrazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-2,1,3-benzothiadiazole-4-sulfonamide
N'-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,N,N'-trimethylbutanediamide
(4S)-1-(2,6-difluoro-3-methoxybenzoyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
2-{2-[3-(trifluoromethyl)phenyl]phenyl}ethan-1-amine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(3-methylphenyl)methyl]amine
2-[(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}piperidin-1-yl)methyl]pyridine
(3S)-4-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
1-(2-chlorophenyl)-2-{[4-(propan-2-yl)pyrimidin-2-yl]amino}ethan-1-ol
(1S,5R)-3-benzyl-6-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperidin-4-amine
(3R,4R)-4-(hydroxymethyl)-1-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]piperidin-3-ol
4-{4-[4-(methoxymethyl)piperidine-1-carbonyl]phenoxy}-N,N-dimethylpiperidine-1-sulfonamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylbenzamide
N-(2-ethoxyphenyl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
2-(2-chloro-4-fluorophenyl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
8-[(2,3-difluorophenyl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-(furan-2-ylmethyl)-N-methylpyridin-2-amine
[1-(4-{4-[4-(pyridin-3-ylmethyl)piperazin-1-yl]piperidin-1-yl}benzoyl)piperidin-3-yl]methanol
1-cyclohexyl-4-[6-(furan-3-yl)pyridine-3-carbonyl]-1,4-diazepane
4-ethyl-3-({1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(1-methyl-1H-imidazol-2-yl)-1-[4-(1H-pyrazol-5-yl)phenyl]-1H-imidazole
N-[(2,4-dimethoxyphenyl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
8-[(4-methanesulfonylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decane
N,1-dimethyl-N-[(3-{[1-(pyridine-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperidin-4-amine
3-[1-(1,3-benzoxazol-2-yl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
ethyl 4-benzyl-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidine-4-carboxylate
4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}morpholine-2-carboxamide
(4aR,7aS)-N,N-dimethyl-4-{[4-(methylsulfanyl)phenyl]methyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridine-3-carboxamide
2-ethyl-5-{2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-6-methyl-3,4-dihydropyrimidin-4-one
{1-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}methanol
ethyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(2-methylprop-2-en-1-yl)amine
2-amino-4-(4-hydroxy-3-methylphenyl)-6-(pyridine-4-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N3-ethyl-N5-[(2-methylphenyl)methyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{[5-(oxan-2-yl)furan-2-yl]methyl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
4-methyl-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(propan-2-yl)pyrimidine-5-carboxamide