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5-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1H-1,2,3-benzotriazole
8-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[4-(4-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]amino}-N,2-dimethylpropanamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
4-(3-phenyl-1H-pyrazol-4-yl)-1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazole
[3-(cyclopropylmethyl)-1-(5-methylthiophene-3-carbonyl)piperidin-3-yl]methanol
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[4-(furan-2-yl)phenyl]-1-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
(1R,7S)-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-3-(3-methylbutyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
methyl (2R,4S)-4-hydroxy-1-(2,4,5-trimethylbenzoyl)piperidine-2-carboxylate
2-{[(3R,5S)-1-[(2-fluorophenyl)methyl]-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]sulfanyl}pyrimidine
N-[(2-fluorophenyl)methyl]-2-{[3-(2-hydroxyphenyl)propyl]amino}acetamide
1-ethyl-5-{[3-(morpholin-4-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[2-(2-hydroxyethoxy)ethyl]quinoxaline-5-carboxamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylpentanamide
6-phenyl-N-(quinolin-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(4-{2-[2-(3-methoxyphenyl)azetidin-1-yl]acetamido}phenyl)-N-methylacetamide
N4-cyclopropyl-7-(2,5-dihydro-1H-pyrrole-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-cyclohexyl-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
3-{[2-(2-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
3-({[(1R)-2-hydroxy-1-phenylethyl]carbamoyl}amino)-4-methyl-N-propylbenzamide
2-(morpholin-4-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
2-(2-methoxyphenyl)-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
4-methyl-3-oxo-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(3-methoxypropyl)-9-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-butyl-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
N-{[7-(3,4-dimethylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
3-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1-(2-methyl-5-sulfamoylphenyl)urea
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methylpyridine-3-carbonitrile
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(prop-2-en-1-yl)acetamide
(2S,4R)-N-(1-benzothiophen-2-ylmethyl)-N-methyl-4-[(4-methylpyrimidin-2-yl)sulfanyl]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
N-[1-(4-chlorophenyl)cyclopropyl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[2-(1,3-benzothiazol-2-yl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
[3-benzyl-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]methanol
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1-[4-(propan-2-yloxy)phenyl]pyrrolidin-2-one
N-(5-methyl-1,3-thiazol-2-yl)-3-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)benzamide
2-(dimethylamino)-1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]ethan-1-one
4-({4-methyl-5-[1-(oxane-4-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
[3-(cyclopropylmethyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl]methanol
2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methylacetamide
3-butyl-4-(thiophen-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{3-oxo-3-[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methyl-N-(oxolan-3-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-benzoyl-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine