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N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
methyl 3-(1-benzothiophen-2-ylmethyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
ethyl 4-[(4-chlorophenyl)methyl]-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidine-4-carboxylate
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
(2E)-1-{3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-phenylprop-2-en-1-one
5-cyclopropyl-N-ethyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
methyl 4-(1H-1,3-benzodiazol-1-yl)pyridine-2-carboxylate
1-phenyl-4-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-pyrazole
dimethyl[1-(1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)ethyl]amine
(3R,5S)-N-[2-(1H-imidazol-4-yl)ethyl]-5-(morpholin-4-ylmethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-(1-acetylpiperidin-4-yl)-1-(4-benzylpiperidin-1-yl)propan-1-one
N,N-dimethyl-4-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]piperazine-1-carboxamide
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1-methyl-4-(pyrrolidin-3-ylmethyl)-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
4-[2-amino-3-cyano-6-(1-methyl-1H-pyrrol-3-yl)pyridin-4-yl]-N-methylbenzene-1-sulfonamide
3-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
ethyl 1-[(3-acetylphenyl)carbamoyl]-3-(2-phenylethyl)piperidine-3-carboxylate
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[(1,3-thiazol-2-yl)carbamoyl]methyl}acetamide
2-{3-methyl-5-[2-(morpholin-4-yl)pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl}acetic acid
N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-pyrazole-3-carboxamide
3-(5-methylthiophen-2-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
1-benzyl-4-(5-ethenylpyridin-2-yl)-1,4-diazepan-6-ol
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-3-(1H-1,2,4-triazol-5-yl)benzamide
{1-[2-(4-fluorophenyl)benzoyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-methoxyphenol
ethyl 5-cyclopentyl-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
5-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(1,3-thiazol-2-yl)piperidine
2-({3-[3-(2-methoxyphenyl)phenyl]-1H-pyrazol-1-yl}methyl)-1,3-thiazole
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-(2-hydroxyethyl)-3-methyl-1-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
5-ethyl-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-(4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
4-fluorophenyl (7S,9aR)-7-[(1R)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-(1-benzothiophen-2-ylmethyl)-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-(dimethylamino)-2-{4-[(2-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}but-3-enamide
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
N-(1,1-dioxo-1λ6-thian-4-yl)-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(furan-2-ylmethyl)(prop-2-yn-1-yl)amine
4-(4-{[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
4-(2H-1,3-benzodioxol-5-yl)-2-[5-(furan-2-yl)-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
3-[(4-fluorophenyl)methyl]-5-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-5-(pyridin-3-yl)imidazolidine-2,4-dione
1-(3-methoxypropyl)-3-{2-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2-oxoethyl}-3-phenylpyrrolidine-2,5-dione
1-{5-methoxy-2-[({[4-(methylsulfanyl)phenyl]methyl}amino)methyl]phenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
3-(4-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid