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2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylacetamide
N,N-dimethyl-3-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyrazin-2-amine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[3-(2-methylphenyl)benzoyl]pyrrolidin-3-yl]methanol
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-methyl-N-(propan-2-yl)acetamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-5-methyl-1,2-oxazole-3-carboxamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
3-benzyl-5-{6-methylimidazo[2,1-b][1,3]thiazol-3-yl}-1H-1,2,4-triazole
N-[3-(2-methoxyphenyl)propyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
5-fluoro-N-[2-methoxy-1-(pyridin-2-yl)ethyl]quinazolin-4-amine
1-benzyl-8-(1H-indol-2-ylmethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({3-[2-(4-fluorophenyl)azetidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-indole
6-ethyl-1,5-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-N-(prop-2-en-1-yl)-1,2-dihydropyridine-3-carboxamide
N-cyclopentyl-5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-(9H-purin-6-yl)pyrrolidin-3-ol
4,5-dimethyl 1-[(3S,5S)-1-[(3,4-difluorophenyl)methyl]-5-[(furan-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-[(2-methoxyethyl)amino]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
3-(4-chlorobenzoyl)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
3-{3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-3,4-dihydroquinazolin-4-one
2-{4-[(2,5-dimethylphenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(2,3-dimethoxyphenyl)methyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-{4-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]piperazin-1-yl}-2,5-dimethylpyrimidine
N-(furan-3-ylmethyl)-N,1-dimethyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
methyl 3-(2-methoxybenzamido)-5-{[3-(3-methoxyphenyl)propanamido]methyl}benzoate
2-ethoxy-3-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]pyridine
2-phenoxy-N-(2-{7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
1-{4-[(2E)-4-methylpent-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
2-{4-[(3,4-difluorophenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
4-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-2,1,3-benzoxadiazole
N-(3-chloro-4-propanamidophenyl)-4-[(prop-2-en-1-yl)amino]benzamide
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyridine-4-carboxamide
6-(2-phenylmorpholin-4-yl)-9H-purine
6-[(3,5-difluorophenyl)methyl]-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
9-methoxy-N-methyl-3-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1,4-diazepan-5-one
(3S,4S)-1-(6-ethyl-5-fluoropyrimidin-4-yl)-4-methylpiperidine-3,4-diol
ethyl 3-benzyl-1-(2,5-dimethoxybenzenesulfonyl)piperidine-3-carboxylate
N-[(2S,4R,6S)-2-benzyl-6-(3-fluoro-5-methylphenyl)oxan-4-yl]acetamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(4-ethylpiperazin-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
2-(4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
7-[ethoxy(phenyl)methyl]-4-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1'-[(5-fluoro-2-methoxyphenyl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
2-chloro-4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]phenol
1-[(3-methylpyridin-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-{1-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}phenol
2-(3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzoyl)-1,2-oxazinane
(3S,4R)-N,N-dimethyl-1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]-4-(propan-2-yl)pyrrolidin-3-amine