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1-{[1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidin-3-yl]methyl}pyrrolidin-2-one
N,N-diethyl-1-(1-{2-[2-(4-fluorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carbonyl)piperidine-3-carboxamide
5-{2-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-3-carboxamide
2-[2,5-dioxo-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-2-ylmethyl)piperidine
3-[(2,3-dimethoxyphenyl)methyl]-5-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
N-[(2R,3R)-1'-cyclopentanecarbonyl-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]acetamide
1-[(3S,4S)-3-[ethyl(methyl)amino]-4-hydroxypyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
(2S,3R)-2-amino-3-hydroxy-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]butan-1-one
3-[(3R,4S)-4-(dimethylamino)-1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl]propan-1-ol
N-{1-[1-(5-chloro-3-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
3-methyl-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)pyridine-2-carboxamide
{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(oxolan-2-ylmethyl)propylamine
3-cyclopropyl-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
2-(5-acetylthiophen-3-yl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
N-[(2R,3R)-1'-{[2-(furan-2-yl)phenyl]methyl}-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(methyl)(quinolin-5-ylmethyl)amine
3-({cyclopropyl[(4-hydroxyphenyl)methyl]amino}methyl)-7-methyl-1,2-dihydroquinolin-2-one
2-cyclopentyl-9-[2-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-chloro-2-propanamidobenzoyl)piperidine-4-carboxylic acid
3-(2-methoxybenzoyl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidine
1-(4,7-dimethylquinazolin-2-yl)-N-[1-(4-methoxyphenyl)ethyl]-N-methylpiperidine-3-carboxamide
3-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}pyrazine-2-carbonitrile
(2S,3R)-3-hydroxy-2-[(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidin-4-yl)formamido]butanamide
(1R,5S,6S)-N,N-dimethyl-3-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
1-(1-methylpiperidin-4-yl)-4-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperazine
(1R,5S,8S)-3-(5,6-dimethylpyrimidin-4-yl)-8-methoxy-3-azabicyclo[3.2.1]octane
(3R,4S)-1-(2,5-dimethylbenzenesulfonyl)-4-propylpyrrolidin-3-amine
N-({7-[3-(4-fluorophenyl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
5-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazine-1-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-(3-methoxypropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
N-(2-methoxyethyl)-1-[1-(thiophene-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-methyl-5-[(2S)-2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-1H-pyrrole-3-carbonitrile
5-chloro-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)thiophene-2-sulfonamide
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
[1-(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)piperidin-2-yl]methanol
3-{[(3-methylpyridin-2-yl)methyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
[(3R,5R)-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
[2-(1H-imidazol-1-yl)ethyl](methyl){[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
(2S)-2-amino-1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
N-cyclopentyl-2,6-difluoro-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzene-1-sulfonamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(diethylamino)acetamide
6-(dimethyl-1,3-thiazole-5-carbonyl)-N-(3,3-diphenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-6-(propan-2-yl)-1H-indole-2-carboxamide
N-[(1S,2R)-2-[(1-acetylpiperidin-4-yl)amino]cyclobutyl]-3-(6-oxo-1,6-dihydropyridazin-3-yl)propanamide
2-hydroxy-S-[3-(piperazine-1-carbonyl)phenyl]-3-(pyrrolidin-1-yl)propane-1-sulfonamido