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N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(4-propyl-1,4-diazepan-1-yl)pyridine-3-carboxamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
methyl 1-ethoxy-8-[(6-methylpyridin-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
ethyl 5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(isoquinolin-5-ylmethyl)-N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
3-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}benzonitrile
4-ethyl-6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyrimidine
2-{1-[(4-methylphenyl)methyl]-4-[(3-methylquinoxalin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-cycloheptyl-6-oxo-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
3-({2-[1-(3-chlorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N,N-dimethyl-2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetamide
[(3R,4R)-1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(4aS,8aR)-6-(2,3-difluorobenzoyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-methyl-5-{1-[5-(6-methyl-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
9-[(3-chloro-2-fluorophenyl)methyl]-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
4-[2-(ethylamino)pyrimidine-5-carbonyl]-1-(2-methylphenyl)piperazin-2-one
dimethyl(3-{2-[1-(pyridin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
N-cyclopropyl-3-{1-[5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carbonyl]piperidin-4-yl}propanamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
1-{9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
(4aS,7aR)-1-(2-butoxyacetyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
7-chloro-N-(1,1-dioxo-1λ6-thiolan-3-yl)-3,5-dimethyl-N-(prop-2-en-1-yl)-1-benzofuran-2-carboxamide
2-methyl-6-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}pyrimidin-4-ol
1-(3-methoxyphenyl)-6-methyl-4-[4-(1H-pyrazol-1-yl)benzoyl]piperazin-2-one
N-[(2-chlorophenyl)methyl]-3-{1-[3-(2-fluorophenyl)propanoyl]piperidin-3-yl}propanamide
2-(4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)pyrazine
2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
8-(4-aminopyrimidin-2-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}azepane
2-(2H-1,3-benzodioxol-5-yl)-N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)acetamide
(3R,5S)-N-butyl-1-[(4-hydroxyphenyl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]piperidine-3-carboxamide
2-[4-(3,4-diethoxyphenyl)-1H-imidazol-2-yl]-4-methoxyphenol
(2R,3R,6R)-5-{imidazo[1,2-a]pyridine-2-carbonyl}-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-methyl-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-methoxy-2-methylpropan-1-one
N-({7-[5-(methoxymethyl)furan-2-carbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenoxypropanamide
2-(2-methyl-1,3-thiazol-4-yl)-N-{1-[(2E)-3-phenylprop-2-en-1-yl]azepan-3-yl}acetamide
[2-(3-methyl-3-phenylpiperidin-1-yl)-1,3-thiazol-4-yl]methanol
[(4-cyclopropyl-5-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-(2-fluoro-5-methylphenyl)-N'-{[2-(1H-imidazol-1-yl)phenyl]methyl}butanediamide
8-(2,2-dimethylpropyl)-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(2-methylphenyl)acetamide
5-methyl-4-{2-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-pyrazol-3-one
4-methyl-5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
2-[1-cyclohexyl-5-(2,3-dihydro-1,4-benzodioxin-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
N,4-dimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-3-(2-oxoimidazolidin-1-yl)benzamide
3-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-2-(methylsulfanyl)pyridine