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3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-[(2,6-difluorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(1-{1-[1-(trifluoromethyl)cyclopropanecarbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
4-{6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrazine-2-carbonyl}morpholine
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[(5-methylfuran-2-yl)methyl]amine
N-[3-(furan-2-yl)propyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]propanamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(5-methyl-1H-pyrazol-1-yl)propanamide
2-{4-[(3,5-difluorophenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N,N-dimethyl-2-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline
7-(morpholin-4-ylmethyl)-4-(2,4,5-trifluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-acetylphenoxy)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
1-(7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
3-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-(3-sulfamoylphenyl)urea
1-[(2-hydroxy-5-methoxyphenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
{4-[4-(trifluoromethyl)pyrimidin-2-yl]-1,4-oxazepan-6-yl}methanol
methyl 3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{2-[1-(2,4,5-trimethylbenzoyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(1-methylpiperidin-4-yl)acetamide
N-benzyl-N,1-dimethyl-5-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,2S)-2-{4-[(3-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}cyclohexan-1-ol
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[4-({1-[4-(morpholin-4-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
1-(cyclohexylmethyl)-3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-3-hydroxypiperidin-2-one
(3E)-1-(4-benzoylpiperazin-1-yl)-4-phenylbut-3-en-1-one
N-{[1-(dimethylamino)cyclohexyl]methyl}-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-fluoro-2-{[2-(2-hydroxyethyl)piperidin-1-yl]methyl}quinolin-4-ol
1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-1,4-diazepan-5-one
2-({3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)phenol
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(morpholin-4-yl)butanamide
7-(furan-2-ylmethyl)-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-[1-(pyridin-3-ylmethyl)piperidin-2-yl]-1H-1,3-benzodiazole
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,3-oxazole-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(prop-2-en-1-yl)amino]piperidin-1-yl}benzamide
1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}isoquinoline
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1H-imidazole-2-carboxamide
1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-4-(2,2,2-trifluoroethyl)piperazine
(3S,4R)-4-(pyridin-3-yl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)pyrrolidine-3-carboxylic acid
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
8-(2-methoxyethyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{[4-(piperidine-1-sulfonyl)-1,4-diazepan-1-yl]methyl}-1H-indole
3-(cyclopropylmethyl)-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
6-[(2-chloro-6-fluorophenyl)methyl]-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(cyclohexylmethyl)-4-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-3-ol
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide