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1-{1-[2-(2-chloro-6-fluorophenyl)acetyl]piperidin-4-yl}-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
N-cyclopentyl-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-{1-[5-(3-acetylphenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-yl}acetamide
1-{[5-chloro-3-methoxy-2-(propan-2-yloxy)phenyl]methyl}pyrrolidin-3-amine
N-(2-methylpropyl)-1-[(1s,4s)-4-[3-(3,4-dimethoxyphenyl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
6-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-N-(propan-2-yl)pyrimidin-4-amine
N-[(3R,4S)-4-cyclopropyl-1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]-2-hydroxyacetamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(3R,4S)-1-(3-hydroxypropyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-methyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-propylacetamide
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(3,4-dimethoxyphenyl)methyl]-N-methylacetamide
2-(4-acetamidopiperidin-1-yl)-2-(4-methoxy-3,5-dimethylphenyl)acetic acid
N-benzyl-1-cyclohexyl-N-[2-(dimethylamino)ethyl]-1H-1,2,3-triazole-4-carboxamide
(4-{[1-(4-methyl-1H-imidazole-2-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
methyl 3-[(3-methoxyphenyl)methyl]-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
3-({2-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
(4aS,7aR)-1-(1-benzofuran-3-carbonyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[(1S,3R)-3-aminocyclopentanecarbonyl]-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
3-[4-(dimethylamino)phenyl]-1-[(3R,4R)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]propan-1-one
3-(2-{[(2,3-dihydro-1H-inden-2-yl)carbamoyl]amino}phenyl)-N-methylpropanamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
1-[3-(3-methoxypropyl)piperidin-1-yl]-2-(4-methylphenyl)ethan-1-one
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
5-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
3-(4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,4-oxazepan-6-yl}methanol
(1R,5R)-6-[3-(4-fluorophenoxy)propyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(2,6-dimethoxyphenyl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
1-[1-(2-hydroxyethyl)-3-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl]-2-methylpropan-1-ol
2-{4-[2-amino-3-cyano-6-(2,2-dimethylcyclopropyl)-5-methylpyridin-4-yl]-2-methoxyphenoxy}acetamide
[(3-cyclohexyl-1H-pyrazol-4-yl)methyl](1H-imidazol-2-ylmethyl)methylamine
N4-methyl-6-(2-methylquinolin-5-yl)pyrimidine-2,4-diamine
5-(5-methyl-2-oxo-5-phenylpiperidin-1-yl)pentanoic acid
3-(1,3-dimethyl-1H-pyrazol-5-yl)-7-ethyl-2,4,5,7-tetraazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene
3-{2-[2-(4-methoxy-2,3,6-trimethylphenyl)-1H-imidazol-1-yl]ethyl}-4-methyl-4H-1,2,4-triazole
N-[2-(3,4-dimethoxyphenyl)ethyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
N-{3-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]phenyl}propanamide
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-(5-oxo-1,4-diazepan-1-yl)pyridine-3-carboxamide
1-{5-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-2-ylmethyl)acetamide
2-(2-fluorophenyl)-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]benzamide
N-[1-(2-phenylethyl)piperidin-3-yl]cyclobutanecarboxamide
N-ethyl-4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-N-phenylbenzamide
3-[(3-chlorophenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-5-(thiophen-2-ylmethyl)-1,2,4-oxadiazole
N-{[2-(2-acetamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
2-cyclopropyl-9-(1H-imidazole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one