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3-[(4aR,7aS)-4-(3-methyl-1H-pyrazole-5-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
(1S,5R)-N-[2-(2-fluorophenyl)ethyl]-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propan-1-one
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2,4-dimethoxybenzamide
3-{5-[2-(4-fluorophenyl)-2-hydroxyacetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-methyl-5-(2-oxo-2-{2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-3,4-dihydropyrimidin-4-one
8-(6-methylpyrimidin-4-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3S,4R)-4-(2-methylphenyl)-1-{[2-(propylamino)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
N-[(2R,3R)-1'-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)methanol
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
(3R,4R)-4-ethyl-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]piperidine-3,4-diol
N-(3-fluorophenyl)-1-(2,3,6-trifluorobenzoyl)piperidin-3-amine
2-[4-(2H-1,3-benzodioxol-5-yl)-3-(methoxymethyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-cyclobutylacetamide
6-{4-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
1-[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-3,3-dimethylbutan-1-one
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
(2S)-2-amino-1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
1-[(4-methoxyphenyl)methyl]-N-[2-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-amino-6-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-4-(oxolan-3-yl)pyridine-3-carbonitrile
2-{2-[2-(2-methoxypyrimidin-5-yl)-1H-imidazol-1-yl]ethyl}-4-methyl-6-(trifluoromethyl)pyrimidine
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(pyridin-2-yl)ethyl]azepan-4-amine
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclobutylacetamide
(1R,5R)-3-(pyrazin-2-yl)-6-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
9-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-{[5-(methoxymethyl)furan-2-yl]methyl}piperazin-2-yl}ethan-1-ol
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(quinolin-6-ylmethyl)acetamide
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-[(4-fluorophenyl)methyl]-N-methylacetamide
4-phenyl-1-[4-(1H-pyrazol-1-yl)butan-2-yl]-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazole
methyl(thiophen-3-ylmethyl)[(3-{[1-(3,4,5-trimethoxybenzoyl)piperidin-4-yl]oxy}phenyl)methyl]amine
3-{3-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-9-methyl-9H-carbazole
5-{3-[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
methyl (2S,4R)-4-(2-fluorobenzamido)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
N-[(2,6-dimethylpyridin-4-yl)methyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-{1-[(2,4-difluorophenyl)methyl]azetidin-3-yl}morpholine
1-(methoxymethyl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]cyclobutane-1-carboxamide
2-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)-N-methylpentanamide
6,8-dimethyl-3-{[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
1'-(1-ethyl-5-oxopyrrolidine-3-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-(1-methylpiperidin-4-yl)pyrimidin-2-amine
1-[(4-methylphenyl)methyl]-4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-2-one
4-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-5-fluoropyrimidin-4-yl}morpholine
4-{[4-(cyclopentyloxy)phenyl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-cyclopentyl-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
(1S,9S)-11-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
(3aS,6aS)-2-(ethanesulfonyl)-5-[(2-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
3-(2-ethylphenoxy)-1-(oxane-2-carbonyl)azetidine
1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine