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5-[(3-fluorophenyl)methyl]-7-({[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
6-[(diethylamino)methyl]-N,N-diethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-methyl-5-{[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}furan-2-carboxamide
N2-[3-(dimethylamino)-2,2-dimethylpropyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
(3aR,6aR)-2-methyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]-5-methyl-1,2-oxazole-3-carboxamide
N-{[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
(3S,4S)-1-[(3-fluoropyridin-4-yl)methyl]-4-(3-methoxyphenyl)piperidin-3-ol
1-[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]-4-(2-methoxyethyl)piperazine
4-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
4-(2-methyl-1H-imidazol-1-yl)-1-[6-(trifluoromethyl)pyridin-2-yl]piperidine-4-carboxylic acid
9-(4-methoxy-2-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(3-fluoro-4-methoxybenzoyl)-2-(2-phenylethyl)morpholine
N4-(azepan-2-ylmethyl)-6-(propan-2-yl)pyrimidine-2,4-diamine
1-(3-fluorobenzoyl)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
5-fluoro-2-[1-(3-phenyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2,6-dimethylquinoline-4-carboxamide
N-(4-fluorophenyl)-1-[2-(morpholin-4-yl)benzoyl]piperidin-3-amine
5-[1-(3-fluorobenzoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
4-benzyl-N-(4-cyano-2-ethylphenyl)-2-(hydroxymethyl)piperazine-1-carboxamide
[5-(5-methyl-1H-indol-3-yl)thiophen-2-yl]methanamine
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]urea
(2R)-2-amino-3-(ethylsulfanyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
1-(1-benzyl-1H-pyrazole-4-carbonyl)-3-(5-fluoro-2-methoxybenzoyl)piperidine
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]propanamide
N-[(6-methylpyridin-2-yl)methyl]-6-[(3-phenoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-hydroxy-3-methyl-N-{2-[4-(oxan-4-yl)morpholin-2-yl]ethyl}benzamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
methyl 2-(azepane-1-sulfonyl)-6-(2,2-dimethylpropyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}but-3-enamide
1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
1-(furan-2-yl)-2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethane-1,2-dione
dimethyl({4-methyl-5-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
5-tert-butyl-N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-1,3,4-oxadiazol-2-amine
N-methyl-N'-(4-methylphenyl)-N-[(3-methylpyridin-2-yl)methyl]propanediamide
N-[(3-methylpyridin-4-yl)methyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,5-dimethylbenzamide
4-methyl-5-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}pyrimidine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
5-[4-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
N-(2-fluoroethyl)-3-{[3-(pyridin-4-yl)propyl]sulfamoyl}benzamide
5-{1-[2-(1,3-thiazol-4-yl)ethyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
N-methyl-N-[2-(oxan-2-yl)ethyl]-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
N-benzyl-5-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}pyrimidin-2-amine
4-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(4-fluorophenyl)-1,4-diazepane
4-(3-hydroxypyridine-2-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide