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N5-cyclooctyl-N3,N3-diethyl-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]acetamide
1-(2-methoxyethyl)-6-oxo-N-[4-(pyridin-2-yl)butyl]piperidine-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-1,3-thiazole-4-carboxamide
methyl 2-[(cyclopropylmethyl)(propyl)sulfamoyl]-6-(pyridin-4-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{2-[2-(trifluoromethyl)morpholine-4-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(3,7-dimethyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-phenyl-1-[1-(pyridin-4-yl)piperidin-4-yl]ethan-1-ol
1-(cyclopropylmethyl)-5-(2,4-dimethoxybenzoyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[4-(2-phenylethyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl]methanol
N-{[5-(4-chlorophenyl)-1,2-oxazol-3-yl]methyl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
11-{[(2,6-difluorophenyl)methyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[(5-acetylthiophen-3-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(2S,4R)-4-(dimethylamino)-1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}pyrrolidine-2-carboxylic acid
1,9-dimethyl-4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(pyridin-2-yl)propanamide
2-(4-chlorophenyl)-4-(5-ethyl-2-methylpyrimidin-4-yl)morpholine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1,2-dimethyl-1H-imidazole-4-sulfonamide
1-cyclopentyl-3-(3-methoxyphenyl)-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
1-methyl-2-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
2-methyl-6-{1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}pyrimidin-4-ol
2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N,N-bis(prop-2-en-1-yl)acetamide
3-cyclohexyl-N-methyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
2-(ethylamino)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]pyrimidine-5-carboxamide
1-(6-methoxypyridin-3-yl)-3-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]urea
1-(3-chlorophenyl)-4-(2-hydroxynaphthalene-1-carbonyl)piperazin-2-one
3-methyl-8-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(2S)-2-amino-3-hydroxy-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
2-({[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-1-(2-methoxyethyl)piperidine-4-carboxamide
2-{[4-(1H-imidazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-propyl-1H-imidazole
2-(4-methyl-1,3-oxazole-5-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-(6-methoxynaphthalene-2-carbonyl)piperidine
1,7-dimethyl-5-[3-methyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-2,4-dione
N-benzyl-4-{2-[(3-methoxyphenyl)carbamoyl]ethyl}piperidine-1-carboxamide
1-(4-chlorophenyl)-5-methyl-4-[4-(methylsulfanyl)benzoyl]piperazin-2-one
1-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]azepane
N-(3-methylphenyl)-N-{2-oxo-2-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethyl}methanesulfonamide
1-{7-[1-(dimethylamino)-2-hydroxypropan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-4-methylpentan-1-one
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
4-(2,6-dimethoxypyridine-3-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3-azaspiro[5.5]undecan-9-amine
3-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
4-(benzyloxy)-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]butan-1-one
(2E)-3-(3-fluorophenyl)-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}prop-2-en-1-one
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
N-[1-(4-methoxyphenyl)propyl]-N-methylimidazo[1,2-a]pyridine-3-carboxamide
8-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
1-cyclopropyl-1-[(4-hydroxy-3-methoxyphenyl)methyl]-3-(1-methyl-1H-indazol-5-yl)urea
1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]piperidin-3-ol