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N-[(2R,3R)-1'-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclopropanecarboxamide
1-methyl-4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidine
3-fluoro-N-{1-[1-(4-methoxy-3-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-(4-fluorophenyl)-N-(pyridin-2-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
8-(3-ethyl-1,2-oxazole-5-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1-methyl-2-oxoimidazolidine-4-carboxamide
N,4-dimethyl-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,3-thiazol-2-amine
1-[2-(1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)piperidin-1-yl]ethan-1-one
methyl 4-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-4-oxobutanoate
1-methyl-4-[(5-propylfuran-2-yl)methyl]piperazine-2-carboxylic acid
5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-N-cycloheptyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(1-cyclopropylethyl)-2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
{3-benzyl-1-[1-(2-methoxyphenyl)piperidin-4-yl]piperidin-3-yl}methanol
3-phenoxy-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
4-[4-(pyrazin-2-yl)piperazin-1-yl]quinazoline
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
1-(2-chlorophenyl)-4-[(4-methoxy-3-{[1-(pyridine-4-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
1-(2-methoxyethyl)-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)piperidin-2-one
3-(cyclopropylmethyl)-1-(3,6-dimethylpyrazin-2-yl)piperidine-3-carboxylic acid
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
(3aS,6aS)-2-[5-(ethoxycarbonyl)pyridin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3,3,3-trifluoropropan-1-one
1-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-2,4-dimethyl-1,4-diazepane
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N,2-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-benzothiazole-5-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[3-(dimethylamino)benzoyl]piperidin-3-yl]propanoic acid
2-{5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-1-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl}acetamide
4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine
N-[(3R,4S)-1-methyl-4-phenylpyrrolidin-3-yl]-4-(2-oxopiperidin-1-yl)butanamide
2-(2-aminoethyl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinazolin-4-amine
(1S,5R)-6-(4-chloro-3-methylbenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(carbamoylmethyl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]piperidine-4-carboxamide
(4aS,8aR)-6-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
methyl 3-(2-cyclopentylacetyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methylbenzamide
N-({4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
N-[(2-methylpyridin-4-yl)methyl]-4-(piperidin-1-yl)butanamide
ethyl 4-(2-methoxyethyl)-1-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]piperidine-4-carboxylate
7-chloro-4-[1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(3-methoxybenzoyl)-4-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
(1R,5R)-6-benzyl-3-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-methyl-2-(morpholin-3-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(pyridin-4-yl)ethan-1-one
N-[3-(4-fluorophenyl)phenyl]-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidine-3-carboxamide
1-[3-(pyridin-4-yl)-5-[1-(pyrrolidin-1-yl)cyclopentyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
5-[1-(4-acetylbenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
1-[2-(cyclohexylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[(3,5-dimethoxyphenyl)methyl]piperidine-4-carboxamide
(1R,2R)-2-(4-{1-[2-(pyrrolidin-1-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)cyclohexan-1-ol