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3-{2-[methyl(2-phenylethyl)amino]ethyl}-8-(1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-({[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}methyl)-5-(hydroxymethyl)-2-methylpyridin-3-ol
14-[4-(propan-2-yl)-1,3-thiazol-2-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-ethyl-2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyridine-4-carboxamide
N-[(3-methoxyphenyl)methyl]-3-[1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl]propanamide
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
N-[(4-hydroxyazepan-4-yl)methyl]-2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzene-1-sulfonamide
7-(cyclopropylmethyl)-2-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(3-hydroxyadamantan-1-yl)ethyl]-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
2-[3-(4-phenoxybenzoyl)piperidin-1-yl]propane-1,3-diol
1-[2-({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-2-one
3-fluoro-N-[1-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
4-(2,5-dimethoxyphenyl)-2-{5-methyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}pyrimidine
4-[4-(4-fluorophenoxy)piperidine-1-carbonyl]-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidine
1-{1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(3-methoxyphenyl)ethan-1-one
5-(3-fluorophenoxymethyl)-N-[(1-hydroxycyclohexyl)methyl]-1H-pyrazole-3-carboxamide
2-{4-[(dimethylamino)methyl]phenyl}-N-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)piperidine-1-carboxamide
4-{[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]methyl}benzoic acid
N-[2-(4-fluorophenyl)-1-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
2-methoxy-N-[2-(thiophene-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[3-(4-fluorophenyl)oxolan-3-yl]methyl})amine
1-(2-ethoxyethyl)-N,3-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-pyrazole-5-carboxamide
(1R,9aR)-1-[(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)methyl]-octahydro-1H-quinolizin-1-ol
(2S,4S)-1-[(3-methylphenyl)methyl]-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazine-2-carboxylic acid
N-ethyl-6-(3-fluorophenyl)-N-[(1R,2R)-2-hydroxycyclohexyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(2-methoxybenzoyl)-1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
2-[benzyl({[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl})amino]ethan-1-ol
4-(2,1,3-benzothiadiazol-5-ylmethyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-amino-4-(oxolan-3-yl)-5H,6H,7H,8H,9H,10H-cycloocta[b]pyridine-3-carbonitrile
2-(5-acetylthiophen-3-yl)-N-[(2,4-difluorophenyl)methyl]acetamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidine-4-carboxamide
N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)-4-phenylbenzamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
5-[(4-chlorophenyl)methyl]-5-{3-oxo-3-[3-(pyridine-3-carbonyl)piperidin-1-yl]propyl}pyrrolidin-2-one
4-{[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-[(3S)-1-benzylpiperidin-3-yl]-1,5-dimethyl-1H-pyrrole-2-carboxamide
4-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-N,N-dimethyl-4-oxobutanamide
1-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-2-one
(3aR,5R,6S,7aS)-2-(quinoline-6-carbonyl)-octahydro-1H-isoindole-5,6-diol
3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole
1-(2,3-dimethoxyphenyl)-2-(furan-2-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-(2,5-dimethoxyphenyl)-2-[4-(morpholin-4-ylmethyl)piperidin-1-yl]acetic acid
N'-(2,5-dimethoxyphenyl)-N-(oxolan-2-ylmethyl)propanediamide
1-[(3-methoxyphenyl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperazine
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}oxolane-2-carboxamide
2-{[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole