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N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-3-(pyrrolidin-3-yl)benzamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-6-(propan-2-yl)pyrimidin-4-amine
(3S,9aR)-8-(3-methylbenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[5-(1-{6-[(propan-2-yl)amino]pyridin-3-yl}-1H-imidazol-2-yl)thiophen-2-yl]prop-2-yn-1-ol
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(piperidin-1-yl)acetamide
N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
3-ethyl-3-(hydroxymethyl)-N-[2-(4-methoxyphenyl)ethyl]piperidine-1-carboxamide
2-(2-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}phenoxy)acetic acid
1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
4-{1-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
ethyl 3-[(3-methoxyphenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxylate
2-methyl-4-(5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)but-3-yn-2-ol
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
[(2S,4R,5R)-4-[({[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}amino)methyl]-5-(2-fluorophenyl)-1-methylpyrrolidin-2-yl]methanol
N-{[7-(1-benzofuran-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
N-[3-(pyridin-3-yloxy)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(2,4-difluorophenoxy)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]acetamide
1-(2-{1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
N-({7-[5-(methoxymethyl)furan-2-carbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
3-[(1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methyl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[(1-benzothiophen-2-ylmethyl)amino]methyl}-N,N-diethylpyridin-2-amine
[1-(1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
4-[(1R,2R)-2-phenylcyclopropanecarbonyl]-7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aS,8aR)-1-(2-phenylethyl)-6-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-{[(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
3-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
2-methoxy-N-(2-methyl-1-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)acetamide
2-methyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]thieno[3,2-d]pyrimidin-4-amine
1-(2-chlorophenyl)-4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
3-phenyl-8-(2-phenylethyl)-1,8-diazaspiro[4.5]decan-2-one
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
N-butyl-5-(2-cyclopentylacetamido)-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
(7S,9aR)-N-benzyl-6,9-dioxo-7-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
4-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}piperazin-2-one
2,6-dimethoxy-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]pyrimidine-4-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2,4,6-trifluorophenyl)acetamide
2-[(1S,5R)-6-[2-(benzyloxy)ethyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-[(2-ethyl-1,3-thiazol-4-yl)methyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
1-(2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}ethyl)imidazolidin-2-one
(2S,4R)-N-cycloheptyl-1-{[4-(2-methylphenyl)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-(3-fluorobenzoyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
(3S,4S)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
4-{[3-(furan-2-yl)-1-phenyl-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiane-1,1-dione
(2S,4S)-4-amino-N-ethyl-1-{[5-(1,2-oxazol-5-yl)furan-2-yl]sulfonyl}pyrrolidine-2-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
3-(2-phenoxyethyl)-8-[(2S)-pyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(2,5-difluorophenyl)pyridine-4-carbonyl]-4-methylpiperazine
3-{1-[1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-N-methylformamido}propanamide
2-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol