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[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
N-methyl-3-(1-methyl-1H-pyrazole-4-amido)-N-phenylazepane-1-carboxamide
N-(3,4-dimethoxyphenyl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-3-amine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
N-[2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]pyrazine-2-carboxamide
2-(oxolane-3-carbonyl)-7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
1-(cyclopropylmethyl)-5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazol-4-yl}pyridine
(1-methyl-1H-imidazol-2-yl)({1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl})methanol
(3S,4S)-1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-4-(morpholin-4-yl)pyrrolidin-3-ol
1-{2-[1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
N,1-dimethyl-N-{[(2R,5S)-5-[(1-methyl-1H-indazol-5-yl)methyl]oxolan-2-yl]methyl}piperidin-4-amine
5-(methoxymethyl)-N-(4-{5-methyl-4-[(3-phenylpropanamido)methyl]-1,3-oxazol-2-yl}phenyl)thiophene-2-carboxamide
4-(1-benzyl-5-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)morpholine
3-{[7-(2-hydroxy-1-phenoxypropan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-6-methyl-4H-chromen-4-one
6-(1-{pyrazolo[1,5-a]pyridine-2-carbonyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
methyl 3-[({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)carbamoyl]propanoate
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(2-oxooxolan-3-yl)-1,2-oxazole-3-carboxamide
2-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
5-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)imidazolidine-2,4-dione
4,6-dimethyl-2-({[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}amino)pyridine-3-carbonitrile
{7-[6-(propan-2-yl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
1-(cyclopropylmethyl)-3-[3-(1-methyl-1H-imidazol-5-yl)phenyl]-1H-pyrazole
2-cyclopropyl-6-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyrimidin-4-ol
4-[4-(2,6-dimethoxybenzoyl)piperazin-1-yl]-2-[(3-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
(2S,4S)-4-(3-chlorobenzamido)-N-(furan-3-ylmethyl)-N,1-dimethylpyrrolidine-2-carboxamide
N-(1-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,5-difluorobenzamide
5-[3-(2-methylphenyl)piperidine-1-carbonyl]quinoxaline
1-[4-({4-[1-(pyridin-3-yl)propan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
2-{2-[4-(1H-pyrazol-1-yl)benzoyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
2-amino-4-(4-methyl-1H-imidazol-5-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-(2-hydroxyethyl)-1-methyl-N-[(5-methylthiophen-2-yl)methyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
N-[(4-methoxynaphthalen-1-yl)methyl]-6-oxo-N-(propan-2-yl)-1,6-dihydropyridine-3-carboxamide
1-[2-(benzylsulfanyl)ethyl]-3-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
N-[2-(4-methoxyphenyl)phenyl]-1-(2-methylpropyl)piperidine-3-carboxamide
2-[4-(6-cyclopropylpyrimidin-4-yl)piperazin-1-yl]benzonitrile
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[3-(pyridin-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
1-(carbamoylmethyl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
5-(1H-indole-5-carbonyl)-1-methyl-N-[3-(morpholin-4-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(propan-2-yl)-6-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]pyrimidin-2-amine
1-(1-cyclohexylpiperidine-4-carbonyl)-4-(1,3-thiazol-2-yl)piperazine
benzyl N-(1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}pyrrolidin-3-yl)carbamate
1-(3-methoxyphenyl)-4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperazine