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2-methyl-5-(propan-2-yl)-N-[2-(pyrrolidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[7-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1-one
1-{[3-(furan-2-yl)phenyl]methyl}-1,4-diazepane-6-carboxylic acid
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
6-methyl-1-{3-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
2-(2,3-dihydro-1H-inden-1-yl)-N-{[4-(dimethylamino)oxan-4-yl]methyl}acetamide
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
12-(2-hydroxybutyl)-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
N-methyl-3-(2-phenylpropyl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,2-oxazole-5-carboxamide
1-[(2,4-difluorophenyl)methyl]-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
1-[(3-methylphenyl)methyl]-4-[6-oxo-1-(3-phenylpropyl)piperidine-3-carbonyl]piperazin-2-one
N-(1-methoxypropan-2-yl)-N-[(2-methylphenyl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
2-[4-carboxy-4-(3-fluorophenoxy)piperidin-1-yl]-6-methylpyridine-3-carboxylic acid
8-(3-phenylbutyl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)acetamide
[(2S,6S)-4-(pyrimidin-2-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyridin-4-ylsulfanyl)acetamide
methyl 3-(2-methylpropanamido)-6-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
2,3-dimethyl-6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoxaline
8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(azetidine-1-carbonyl)-N-[1-(4-fluorophenyl)ethyl]-N-methylbenzene-1-sulfonamide
2-(dimethylamino)-N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(3-methylphenyl)acetamide
4-methoxy-2-({4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)-3,5-dimethylpyridine
N-(cyclopropylmethyl)-3-(3-hydroxy-3-methylbutyl)-N-propylbenzamide
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-[3-(morpholin-4-yl)propyl]-1,4-diazepane
methyl 3-{[1-(cyclopropylmethyl)-5-(2,6-difluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-[1-(3-phenylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
4-[4-(4-fluorophenyl)-4-oxobutyl]-1-(2-methoxyphenyl)piperazin-2-one
7-(1-benzothiophen-3-yl)-9-methoxy-4-(3-methyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[4-(4-chlorophenyl)butanoyl]piperazine-1-sulfonamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(2H-1,3-benzodioxol-5-ylmethyl)-N-[2-(3-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
3-[3-methyl-5-(quinolin-4-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-[(2R,3R)-1'-[(3-ethoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
5-[(4-fluorophenyl)methyl]-3-(oxolan-3-yl)-5-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
(1R,3S)-3-({3-[(4-chlorophenyl)sulfanyl]propyl}carbamoyl)cyclopentane-1-carboxylic acid
2-{[(3S,5S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]sulfanyl}-4-methylpyrimidine
6-fluoro-2-({[1-(6-methylpyridin-2-yl)propan-2-yl]amino}methyl)quinolin-4-ol
2-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}-5-(pyrrolidine-1-carbonyl)pyridine
N-{[7-(3-cyclopentylpropanoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-2-yl)acetamide
1-cyclopropyl-3-(4-methoxyphenyl)-3-[2-oxo-2-(3-propanoylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N3-tert-butyl-N5-[(2-methoxyphenyl)methyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(4-fluorophenyl)-4-[3-(5-methylfuran-2-yl)benzoyl]piperazine
(2S)-3-[(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]propane-1,2-diol
(3aS,6aR)-5-(3,6-dimethylpyrazin-2-yl)-3-[3-(4-fluorophenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-oxoacetamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
1-methyl-N-{2-[4-(propan-2-yl)morpholin-2-yl]ethyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-2-[4-(3-methyl-1,2-oxazole-5-carbonyl)morpholin-3-yl]-N-[2-(pyridin-2-yl)ethyl]acetamide
2-{[4-(2,4-difluorobenzoyl)-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl]oxy}-N,N-diethylacetamide