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1-cyclopentyl-3-(3-fluorophenyl)-3-{2-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
1-[(1S,5R)-6-(4-methoxybenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
methyl (2S)-3-methyl-2-{[1-(3-phenylpropyl)-1H-1,2,3-triazol-4-yl]formamido}butanoate
2-(4-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}piperidine-1-carbonyl)pyridine
(2E)-3-(4-methoxyphenyl)-N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)prop-2-enamide
3-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
4-{4-[2-(hydroxymethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
(1S,5R)-6-cyclopentanecarbonyl-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
methyl (2S)-2-phenyl-2-({1-[3-(4-phenylbutanamido)phenyl]piperidin-4-yl}amino)acetate
propan-2-yl 2-(4-{2-amino-6-oxo-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-8-yl}phenoxy)acetate
3-(carbamoylamino)-N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]propanamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
2-[1-(1-methylpiperidin-4-yl)pyrrolidin-3-yl]benzoic acid
4-[4-(3-chlorophenyl)-1H-1,2,3-triazol-1-yl]-1-(oxolan-3-ylmethyl)piperidine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[1-(3-fluorophenyl)propan-2-yl]amine
9-(1-benzyl-5-methyl-1H-1,2,3-triazole-4-carbonyl)-3-methyl-3,9-diazaspiro[5.6]dodecane
ethyl 3-[(2-methylphenyl)methyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-3-carboxylate
3-amino-2-hydroxy-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-[4-(2-methoxypyridine-3-carbonyl)morpholine-2-carbonyl]-4-methyl-1,4-diazepane
(1R,9aR)-1-[2-(pyrrolidine-1-carbonyl)phenoxymethyl]-octahydro-1H-quinolizine
4-(3-hydroxy-3-methylbutyl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]benzamide
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-oxazole-3-carboxamide
2-[3-(2-fluorophenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
N-[(3-fluorophenyl)methyl]-3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carboxamide
[(2E)-3,7-dimethylocta-2,6-dien-1-yl][3-(pyridin-4-yl)propyl]amine
[(1-cyclopentylpiperidin-4-yl)methyl][(2,5-dimethoxyphenyl)methyl](pyridin-3-ylmethyl)amine
N-(4-chloro-2-fluorophenyl)-4-(2-methoxyphenoxy)piperidine-1-carboxamide
1-(4-{4-[(3-aminopropyl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(2-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-acetyl-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)piperidine-4-carboxamide
methyl 3-acetamido-1-ethyl-5-{[1-(2-fluorophenyl)propan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(2-ethoxyacetyl)-1-(3-methoxyphenyl)piperazin-2-one
N-[(3S,4R)-1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
4-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]-1,4-oxazepan-6-ol
1-(benzenesulfonyl)-4-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperazine
1-(2-cyclobutylacetyl)-4-(furan-2-ylmethyl)-1,4-diazepane-6-carboxylic acid
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
8-[(2-chloro-6-fluorophenyl)methyl]-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[3-benzyl-1-(quinolin-2-ylmethyl)piperidin-3-yl]methanol
N-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-3-(2-methylphenyl)-3-phenylpropanamide
N-(3-chlorophenyl)-4-[4-(piperazin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
(2R)-2-cyclohexyl-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-hydroxyacetamide
6-hydroxy-1-(pyridin-3-ylmethyl)-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-1,4-diazepan-2-one
3-benzyl-6-(1,4-dioxan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
7-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(1-cyclopentylpiperidin-3-yl)methyl]-1-methyl-N-[2-(piperidin-1-yl)ethyl]-1H-pyrrole-2-carboxamide
5-fluoro-3-[(4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)methyl]-1H-indole
1-[4-oxo-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(pyrrolidin-1-yl)ethane-1,2-dione
7-(1-benzofuran-2-sulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(2-methoxyphenoxy)-1-[3-(methylsulfanyl)propanoyl]piperidine-4-carboxylic acid