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({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)[(3,4-dimethoxyphenyl)methyl]methylamine
N-methyl-2-(piperidin-1-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]acetamide
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[(4-methylphenyl)methyl]piperidine-3-carboxamide
6-[(4-methoxy-3-methylphenyl)methyl]-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1-[(2-chlorophenyl)methyl]-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[5-(2,6-dimethylquinolin-3-yl)-3-methyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperidin-3-yl)methanol
N-(pentan-3-yl)-1-(pyridin-3-ylmethyl)piperidin-3-amine
4-oxo-4-[4-(quinolin-3-yl)phenyl]butanoic acid
4-(2-ethylpyridine-4-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
1-(2-ethylbutyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-[(3R,5S)-1-cyclopropanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
4-(hydroxymethyl)-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}azepan-4-ol
N-benzyl-5-methoxy-N-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
(2E)-1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-3-(thiophen-2-yl)prop-2-en-1-one
2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-methylthiophene-2-carboxamide
4-(2-{1-[(3-chloro-4-methoxyphenyl)methyl]piperidin-2-yl}ethyl)morpholine
4-(pyrrolidine-1-carbonyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzene-1-sulfonamide
6-(4-fluorophenyl)-7-methyl-8-oxo-N-[(1s,4s)-4-aminocyclohexyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(1-benzothiophen-2-ylmethyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(1,4-dioxan-2-ylmethyl)(methyl){[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
3-(2,2-diethylcyclopropanecarbonyl)-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3S,4S)-1-[(E)-2-phenylethenesulfonyl]piperidine-3,4-diol
1-methyl-N-[(1-methylpiperidin-4-yl)methyl]-6-oxo-N-(2-phenylethyl)-1,6-dihydropyridazine-3-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(pyridin-3-yl)propan-2-yl]benzamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[3-(5-methylfuran-2-yl)butyl]piperazine
1-(5-propyl-1,3,4-oxadiazol-2-yl)-4-(pyrrolidin-1-yl)piperidine
(1R,3S)-3-ethoxy-7-(1-phenylpiperidin-4-yl)-7-azaspiro[3.5]nonan-1-ol
{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[1-(pyridin-3-yl)propan-2-yl]amine
ethyl 4-[1-(thiophene-3-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
4-(5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-1,4-diazepane-1-carbaldehyde
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
5-tert-butyl-4-{[2-(furan-2-yl)azepan-1-yl]methyl}furan-2-carboxamide
1,3-dimethyl-5-{[(6-methyl-2-propylpyrimidin-4-yl)amino]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-methyl-1-{1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]azetidin-3-yl}piperidine
2-benzyl-8-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,8-diazaspiro[5.5]undecane
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}-1H-indole
7,8-dimethyl-4-(4-methylpiperidine-1-carbonyl)-2-(pyrimidin-5-yl)quinoline
[3-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-2,4,6-trimethylphenyl]methyl acetate
2-{3-[3-(2,6-dimethylpyridin-4-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N-ethyl-N-methyl-4-(3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanoyl)morpholine-2-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl})amine
4-[(2-methylprop-2-en-1-yl)oxy]-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
1-(2,4-difluorobenzoyl)-2-(3-fluorophenyl)piperidine
N-methyl-6-phenyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyridazin-3-amine
1-cyclopentyl-5-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}piperidin-2-one
2-{[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]methyl}-1,4-dimethylpiperazine