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3,5-dimethyl-4-oxo-N-[2-(1H-1,2,4-triazol-1-yl)propyl]-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-[2-(dimethylcarbamoyl)-1-benzothiophen-5-yl]-2-(ethoxymethyl)pyrrolidine-1-carboxamide
3-{[3-(ethoxymethyl)-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
7-(5-methylthiophen-2-yl)-4-(1,3-thiazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
ethyl 1-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperidine-3-carboxylate
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-[1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
N-[4-fluoro-3-(methylcarbamoyl)phenyl]-2-methyl-4-(2-methylphenyl)piperazine-1-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
4-(1H-pyrazol-1-yl)-1-[2-(pyridin-3-yloxy)acetyl]piperidine-4-carboxylic acid
3-[methyl({3-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-3-oxopropyl})amino]-1λ6-thiolane-1,1-dione
5-(2-chloro-4-methoxyphenoxymethyl)-3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,2-oxazole
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-(thiolan-3-yl)acetamide
2-(pyrrolidin-1-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
1-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}piperidin-4-ol
2-{4-[(5-cyclopentylthiophen-2-yl)methyl]morpholin-3-yl}-1-(pyrrolidin-1-yl)ethan-1-one
1-[4-(quinolin-3-yl)phenyl]ethan-1-ol
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methoxyphenyl)methyl]acetamide
N-[(1-methylpiperidin-3-yl)methyl]-3-(methylsulfanyl)-N-(2-phenylethyl)propanamide
1-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2,2-dimethylpropan-1-one
(2S)-N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-2-hydroxy-N-(2-hydroxyethyl)propanamide
6-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}pyridine-2-carboxylic acid
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-ol
1-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-4-[2-(4-chloro-1H-pyrazol-1-yl)acetamido]-N-ethyl-1-(3-hydroxypropanoyl)pyrrolidine-2-carboxamide
5-butyl-1-(3-phenylphenyl)-4-(pyrazine-2-carbonyl)piperazin-2-one
8-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
methyl (2S)-2-({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)-3-phenylpropanoate
7-fluoro-N-[1-(methoxymethyl)cyclopentyl]-2-methylquinoline-4-carboxamide
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-phenylpropanamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
3-[3-(3-chlorophenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]benzonitrile
methyl 3-[(3-chlorophenyl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl 4-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}benzoate
4-methyl-2-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-6-(trifluoromethyl)pyrimidine
2-cyclopropyl-4-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidine-1-carbonyl}quinoline
3-(diphenylmethyl)-N-(2-methoxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N,N-dimethyl-5-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
4-(2,8-dimethylquinoline-3-carbonyl)-1-(3-methoxyphenyl)piperazin-2-one
4-{1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]piperidin-3-yl}benzoic acid
1,4,6-trimethyl-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
[(1-ethyl-1H-pyrazol-4-yl)methyl](oxolan-3-ylmethyl)(propan-2-yl)amine
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(2,2-diethylcyclopropanecarbonyl)piperidine
2-chloro-4,5-difluoro-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)benzamide
3-(2,3-dihydro-1H-inden-2-yl)-5-{1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
1-{2-[(4-ethylpiperazin-1-yl)methyl]-5-methoxyphenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
3-{[(5-methyl-1,2-oxazol-3-yl)formamido]methyl}-N-(2-phenylphenyl)piperidine-1-carboxamide
1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione