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(1R,4S)-2-{2-[3-(2-methylphenoxy)azetidin-1-yl]pyridine-3-carbonyl}-2-azabicyclo[2.2.1]heptane
ethyl 1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-2-carboxylate
3-(1-ethyl-1H-imidazol-2-yl)-1-(3-phenylpropyl)piperidine
2-{4-[1-(2,3-dimethylphenyl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(1H-imidazol-2-ylmethyl)piperidine-4-carboxylic acid
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(1H-pyrazol-1-yl)benzamide
{[5-(methoxymethyl)furan-2-yl]methyl}({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
5-{[(3-methoxypropyl)amino]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-[1-(cyclohexylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-(2-hydroxy-2-phenylethyl)-N-methylacetamide
4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)propyl]furan-2-carboxamide
N-ethyl-2-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]piperidine-3-carboxamide
6-fluoro-2-{[methyl({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}quinolin-4-ol
(3S,4S)-1-[(2-hydroxy-3,5-dimethylphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
(2S)-N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-acetamido-4-methylpentanamide
(1R,5R)-N,N-dimethyl-6-[2-(3-methylphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[3-(1H-imidazol-1-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
5-(but-3-en-1-yl)-3-(2,6-dimethoxyphenyl)-1,2,4-oxadiazole
1-cyclopentyl-3-(2-methoxyphenyl)-3-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2-[4-(hydroxymethyl)phenyl]-2-[4-(2-methoxyphenoxy)piperidin-1-yl]acetic acid
methyl 4-{[3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
3-{[1-butyl-3-(1H-indol-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
1-(dimethylamino)-2-{4-[(2,4-dimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
(2R)-2-[5-(2-fluoro-4,5-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propanamide
8-{2-[ethyl(methyl)amino]acetyl}-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(4-fluorophenyl)piperidin-1-yl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(pyridin-4-ylmethyl)acetamide
N-(1-methanesulfonylpiperidin-4-yl)-4-(1H-pyrazol-3-yl)benzamide
6-fluoro-2-oxo-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
N-[4-(4-{[(2,4-difluorophenyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)furan-2-carboxamide
N-cyclopropyl-4-{[(1-ethylpyrrolidin-3-yl)methyl](methyl)sulfamoyl}benzamide
(4aS,8aR)-6-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-phenylethan-1-one
4-(azonan-1-yl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyridine-2-carboxamide
(2R)-2-amino-N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-2-phenylacetamide
2-(ethylsulfanyl)-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]propanamide
8-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-fluoro-N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)benzamide
3-(2,3-dihydro-1H-inden-2-yl)-5-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
N-{2-methyl-3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenyl}oxolane-2-carboxamide
methyl 3-[({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)carbamoyl]benzoate
ethyl 4-[6-methyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carbonyl]piperazine-1-carboxylate
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1-(pyrrolidin-1-yl)cyclohexane-1-carboxamide
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-(thiophen-3-ylmethyl)benzamide
2-cyclopropanecarbonyl-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(4aS,7aR)-1-(6-aminopyridine-3-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-N-(propan-2-yl)pyrimidin-2-amine