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N-[(2R)-1-hydroxybutan-2-yl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
7-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl 2-{[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
N-[(2R)-pyrrolidin-2-ylmethyl]-2-(4H-1,2,4-triazol-4-yl)benzamide
4-cyclopentyl-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
1-(2,6-dimethylpyrimidine-4-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
methyl 1-({3-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperidine-4-carboxylate
(2S)-2-amino-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}pentan-1-one
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
4-[2-methyl-2-(morpholin-4-yl)propyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-4-yl)piperazine
5-({4-ethyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-2-(2-methoxyphenyl)-1,3-thiazole
1-{2-methyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-5-phenylpentane-1,5-dione
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[2-(naphthalen-2-yl)ethyl]piperidin-4-amine
N-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-{1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidin-4-yl}piperidin-3-ol
3-(pyrrolidin-1-yl)-1-(thian-4-yl)piperidine
(2S,4S)-1-({4-[2-(dimethylamino)ethoxy]phenyl}methyl)-4-acetamido-N-ethylpyrrolidine-2-carboxamide
1-{7-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4-methylpentan-1-one
2-(cyclopropylmethyl)-9-(6-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
7-{[4-(propan-2-yl)phenyl]methyl}-2-[3-(1H-pyrazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}benzoic acid
(2S,4S)-1-cyclopentyl-N-ethyl-4-(3-hydroxy-2-methylbenzamido)pyrrolidine-2-carboxamide
5-methyl-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1H-pyrazole-3-carboxamide
4-[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-1-(4-fluorophenyl)butan-1-one
4-[(2S)-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidine-2-carbonyl]morpholine
1-(2-methoxyphenyl)-4-[2-(1H-pyrrol-1-yl)butanoyl]piperazin-2-one
(4aR,7aS)-1-methyl-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-ethyl-3-{2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-oxoethyl}piperazin-2-one
3-ethyl-8-(6-oxopiperazine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-methoxyethyl)-1-{1-[3-(trifluoromethyl)benzoyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
3-(azepane-1-carbonyl)-N-(2-methoxyethyl)-N-methyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
S-[2-(furan-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-hydroxybutane-1-sulfonamido
1,3-dimethyl-4-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperazin-2-one
4-methoxy-2-{[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]methyl}phenol
N,1-dimethyl-6-propyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 2-(3-{2-[(4-fluoro-2-methylphenyl)carbamoyl]ethyl}piperidine-1-carbonyl)benzoate
2-methoxy-5-{4-phenyl-1-[2-(piperidin-1-yl)ethyl]-1H-imidazol-5-yl}pyrimidine
1-(cyclobutylmethyl)-3-hydroxy-3-({methyl[(3-methyl-1H-indol-2-yl)methyl]amino}methyl)piperidin-2-one
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypropan-1-one
3-{2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-(1-methyl-6-oxopiperidin-3-yl)benzamide
1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N,N-diethylpiperidine-4-carboxamide
(3S,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-amine
1-(4-{[(2R,5S)-5-[(3,4-difluorophenyl)methyl]oxolan-2-yl]methyl}piperazin-1-yl)ethan-1-one
N-(2-methoxyethyl)-2-methyl-N-(1-methylpiperidin-4-yl)-6-(piperidin-3-yl)pyrimidin-4-amine
N4-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-6-(propan-2-yl)pyrimidine-2,4-diamine