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3-{1-[5-(2-chlorophenyl)furan-2-carbonyl]pyrrolidin-2-yl}-5-methyl-1,2-oxazole
4-(2-methoxybenzoyl)-7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{5-[2-(propan-2-yloxy)phenyl]pyridin-2-yl}acetamide
3-ethyl-5-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1,2-oxazole-4-carboxamide
4-phenyl-N-[3-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]butanamide
1-benzyl-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
4-(3-methyl-1H-1,2,4-triazol-5-yl)-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine
methyl 3-methyl-4-{[4-(oxan-4-yl)piperazine-1-carbonyl]amino}benzoate
2-[cycloheptyl(ethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-(3-{4-[(1-propylpiperidin-4-yl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
1-(5-fluoro-2-methylbenzoyl)-3-(3-methoxypropyl)piperidine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1,2,3,4-tetrahydroquinoline-8-carboxamide
N5,N5-dimethyl-N6-{[1-(morpholin-4-yl)cyclohexyl]methyl}-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
2-({[(3R,4R)-1-[(2,3-difluorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-ethoxy-3-{[5-(5-methylfuran-2-yl)-1,2,4-triazin-3-yl]amino}propan-2-ol
5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrazin-2-ol
N-[(1-cyclopentylpiperidin-3-yl)methyl]-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-N-propyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}propan-1-one
N,N,1-trimethyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecane-4-sulfonamide
2-[4-(3,5-difluoropyridine-2-carbonyl)piperazin-1-yl]-N-ethylacetamide
6-(methoxymethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-methyl-N-(pyridin-2-ylmethyl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
5-fluoro-2-(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-2-yl)-1H-1,3-benzodiazole
N-(1-{[4-(2-phenylethoxy)phenyl]methyl}piperidin-4-yl)acetamide
N'-cyclooctyl-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)butanediamide
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-(2-phenylindolizin-3-yl)ethane-1,2-dione
1-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
5-phenyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
4-[3-(3-hydroxy-3-methylbutyl)benzoyl]-N,N-dimethylpiperazine-1-carboxamide
(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)(pyridin-2-ylmethyl)amine
2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-5-methoxy-1-methyl-1H-indole
3-methyl-1-(1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)butan-1-one
2-(2,5-dimethylphenoxy)-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]propanamide
N-[2-(4-methoxyphenyl)ethyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
7-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
[(3R,4R)-1-[4-(2-methylpropyl)benzoyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-methyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]benzamide
methyl 4-(4-{[(2S)-2-carbamoylpyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
3-ethyl-4-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-1-methylpiperazin-2-one
1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
(2S,4S)-4-(4-{[(4-fluoro-3-methylphenyl)formamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
5-cyclobutanecarbonyl-1'-(pyridazine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[4-(3-methylphenoxy)piperidine-1-carbonyl]benzonitrile
2-(1-ethylpiperidin-4-yl)-1-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]ethan-1-one
1-ethyl-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(6-fluoropyridin-3-yl)-3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
4-methyl-5-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-thiazole