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3-{2-[5-(2-fluorophenyl)furan-2-yl]-1H-imidazol-1-yl}propan-1-ol
methyl (2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-4-[(2-hydroxyethyl)(methyl)carbamoyl]-1-methylpyrrolidine-2-carboxylate
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidine-2-carboxamide
2-(3-fluorophenoxymethyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
3-[(2,6-difluorophenyl)methyl]-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-(2-methoxyethyl)-8-{[4-(methylsulfanyl)phenyl]methyl}-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 2-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1,3-oxazole-4-carboxylate
4-{3-[4-(cyclopentylmethyl)piperazine-1-carbonyl]phenyl}phenol
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methylthian-4-amine
3-fluoro-4-methoxy-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-methyl-6-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)pyrimidin-4-ol
2-{1-[(2-fluorophenyl)methyl]-4-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1H-1,2,3-triazole
(4aS,7aR)-1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[(3,4-dimethoxyphenyl)methyl]-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-methoxy-4-(2-methoxybenzoyl)-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl](benzylsulfamoyl)amine
1-cyclopropyl-4-[3-(2-methylpropyl)-1-(naphthalen-1-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
methyl N-{[(2S,4S)-4-fluoro-1-[2-(pyridin-4-yl)acetyl]pyrrolidin-2-yl]methyl}carbamate
1-({5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
N3-(1-benzylpiperidin-4-yl)-1-cyclopentyl-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
6-chloro-3-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)-4H-chromen-4-one
4-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
4-(4-methoxypiperidin-1-yl)-7-(pyrazin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
1-[(4-fluorophenyl)methyl]-4-(1H-imidazol-2-ylmethyl)-1,4-diazepane
(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
3-(2-methoxyphenyl)-N-[(5-methylpyrazin-2-yl)methyl]benzamide
2-(cyclopropylmethyl)-9-(4-fluoro-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperidine-4-carbonyl)morpholine
3,5-dichloro-N-[2-(1H-imidazol-4-yl)ethyl]-4-(prop-2-en-1-yloxy)benzamide
2-acetyl-8-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[1-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethyl]morpholine
N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
2-{1-cyclopentyl-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(1S,5R)-6-(4-methoxy-3-methylbenzoyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-3-(1,3,4-thiadiazol-2-yl)-1-(thiophen-3-ylmethyl)urea
(1S,6R)-N-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-2-(morpholin-3-yl)acetamide
2-[4-(5-fluoro-1-methyl-1H-indole-2-carbonyl)-1-(furan-2-ylmethyl)piperazin-2-yl]ethan-1-ol
2-(2-ethyl-1H-imidazol-1-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
2-amino-1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-methylpropan-1-one
2-[(5-methylpyrazin-2-yl)methyl]-8-(oxan-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-chloro-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
3-(3-methoxyphenyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-(2-{4-[(2-methoxy-2-phenylacetamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-2,5-dimethylfuran-3-carboxamide
2-(naphthalen-1-yl)-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
1-[(4-methoxyphenyl)methyl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-1,2,3-triazole-4-carboxamide