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ethyl 4-[1-(3-methylbutyl)-2,4-dioxo-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]piperidine-1-carboxylate
2-(2-hydroxyphenoxy)-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
3-[(2,3-dimethoxyphenyl)methyl]-5-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
2-(4-ethylpiperazin-1-yl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
4-(5-tert-butyl-1H-pyrazol-3-yl)-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1H-1,2,3-triazole
1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-(oxan-4-ylmethyl)-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
N-(2-{[6-(methoxymethyl)pyrimidin-4-yl]amino}ethyl)pyridine-3-carboxamide
6,7-dimethoxy-1-methyl-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
1-(3-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-3-oxopropyl)azepan-2-one
ethyl[2-(1H-pyrazol-1-yl)ethyl](quinolin-4-ylmethyl)amine
N-(2-{7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
(2S)-2-[1-(2-methylphenyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]pyrrolidine-1-carboxamide
3-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl){[4-(trifluoromethoxy)phenyl]methyl}amine
methyl 3-(2-methoxy-2-phenylacetyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]urea
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole
N-tert-butyl-2-(4-{[3-(hydroxymethyl)-4-methylpiperazin-1-yl]methyl}phenoxy)acetamide
3-{1-[3-(2-chlorophenyl)propanoyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
4-methoxy-N-[2-(3-methoxyphenyl)ethyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
4-fluoro-N-(2-{7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2-(3-chlorophenoxy)-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}propan-1-one
4-[(4-fluorophenyl)methyl]-3-{2-[4-(2-methoxyethoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
3-chloro-6-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyridine-2-carboxylic acid
1-(2-methoxyphenyl)-2,2-dimethyl-4-(1H-pyrazole-3-carbonyl)piperazine
N-(2-ethoxyphenyl)-N'-ethyl-N'-(oxan-4-ylmethyl)propanediamide
N-({7-[3-(4-methoxyphenyl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
2-[(1-cyclobutanecarbonylpiperidin-4-yl)formamido]-2-phenylacetic acid
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidin-4-ol
(3S)-3-benzyl-4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazin-2-one
(2S,4R)-N-[2-(3-chlorophenyl)ethyl]-1-[(3-methylthiophen-2-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-3-(4-phenylbenzoyl)piperidine
4-[5-(5-methyl-1H-pyrazole-3-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
4-fluoro-N-{2-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzamide
N-(1-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
methyl 1-(2-methoxyethyl)-3-(3-phenylpropanamido)-5-({[3-(trifluoromethyl)phenyl]methyl}amino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-acetyl-N-methyl-N-(oxolan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(2-hydroxyethyl)amino]methyl}piperidin-2-one
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-chloro-6-methoxy-4-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
3-(pentan-2-yl)-8-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(2-chlorophenyl)methyl]-7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2,3-dihydro-1H-indene-2-carboxamide
N3-(1-benzylpyrrolidin-3-yl)-N5-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(azepan-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
[3-(2-methylpropyl)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-3-yl]methanol
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one