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(4aS,7aR)-1-(3-ethoxypropanoyl)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-methoxy-1,2-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-indole-3-carboxamide
(1-methyl-1H-imidazol-2-yl)(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
4-[(4-methylthiophen-2-yl)sulfonyl]-2-(2-phenylethyl)morpholine
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(2-methoxyphenyl)propanamide
1-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
2-{3-cyclopentyl-5-[1-(4-oxo-3,4-dihydroquinazolin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
3-{[(2,3-dimethyl-1H-indol-7-yl)methyl](methyl)amino}-N-methylpropanamide
N-[1-({[2-(methylsulfanyl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-phenoxyacetamide
2-(2-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-4-(pyridin-2-yl)phenoxy)acetic acid
9-(2-methoxyethyl)-1-methyl-4-[6-(trifluoromethyl)pyridin-2-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(2-benzyl-5-oxopyrrolidin-2-yl)-N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]propanamide
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-2-cyclopentyl-N-(oxolan-2-ylmethyl)acetamide
5-fluoro-2-[(2-methoxyphenyl)methyl]-1-[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
4-(2-methyl-1,3-thiazole-5-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[(4-hydroxyphenyl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2-methoxyethyl)({[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl})methylamine
[(1-cyclohexylpiperidin-3-yl)methyl][(3-phenyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)amine
2-(dimethylamino)-1-(4-ethoxypiperidin-1-yl)-2-(4-fluorophenyl)ethan-1-one
1-(2-methoxy-4-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-2-carboxylic acid
1-(3-chloro-4-ethoxyphenyl)-3-[1-(furan-2-ylmethyl)piperidin-4-yl]urea
(4aS,8aR)-6-(2,3-dihydro-1H-inden-2-yl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(2-fluorophenyl)ethan-1-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-(2,2,2-trifluoroethyl)acetamide
N-cyclopropyl-3-[1-(4-phenylbenzoyl)piperidin-4-yl]propanamide
4-(cyclopropylmethyl)-1-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(3aR,6aR)-2-cyclohexyl-5-(6-ethyl-5-fluoropyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2R,3R,6R)-5-(3-methoxypropyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2-fluorophenyl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
3-[1-(adamantan-1-yl)piperidin-3-yl]-N-(2-fluorophenyl)propanamide
(2E)-N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(4-methoxyphenyl)prop-2-enamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[3-(1H-pyrazol-1-yl)propyl]amine
4-[(6-chloro-2H-chromen-3-yl)methyl]piperazine-1-sulfonamide
benzyl({[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
4-(2-ethylpyrimidine-5-carbonyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
3-(2-ethyl-1H-imidazol-1-yl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]propanamide
1-{2-[2,5-dioxo-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]acetyl}piperidine-3-carboxamide
[1-({1-[(2,3-dimethyl-1H-indol-7-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
2-{1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl}-6-chloro-1H-1,3-benzodiazole
N,N-dimethyl-5-{[(1-phenylcyclopentyl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-{4-[(6-chloropyridin-3-yl)methyl]morpholin-2-yl}ethyl)azetidine-3-carboxamide
2-[4-(adamantan-1-yl)piperazin-1-yl]acetic acid
N-[(3-fluorophenyl)methyl]-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-[1-(furan-2-yl)ethyl]acetamide
methyl({[5-(oxolan-2-yl)thiophen-2-yl]methyl})[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-[2-(azepan-1-yl)-2-phenylethyl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
2-methyl-8-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
N-(2-methyl-1-{7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)pyridine-2-carboxamide
(1S,5R)-3-[3-(3-methoxyquinoxalin-2-yl)propanoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one