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methyl 2-(2-carbamoylethyl)-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl 5-{4-[(methylcarbamoyl)amino]benzenesulfonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
[(3R,4S)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
5-{5-[2-(benzyloxy)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-methyl-1,2-oxazole
4-(5-ethyl-4-phenyl-1H-imidazol-2-yl)-1-(propan-2-yl)pyrrolidin-2-one
(4aS,8aR)-1-(4-hydroxybutyl)-6-(pyrrolidine-1-sulfonyl)-decahydro-1,6-naphthyridin-2-one
{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}[(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
methyl({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}){[2-(trifluoromethyl)phenyl]methyl}amine
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]pyridin-2-amine
5-({[1-(2-methoxyphenyl)ethyl](methyl)amino}methyl)pyrimidin-2-amine
(2S,4R)-4-hydroxy-1-[2-(2,3,6-trimethylphenoxy)acetyl]pyrrolidine-2-carboxylic acid
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[2-(propan-2-yl)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methanol
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
[(4-methanesulfonylphenyl)methyl](2-methylpropyl)(pyridin-2-ylmethyl)amine
2-(4-methyl-1H-pyrazol-1-yl)-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]propanamide
1-(2-methylpyridin-4-yl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,4-diazepane
5-({2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-(2-fluoro-4-methylbenzoyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N-(1H-indazol-6-yl)-2-[4-(2-phenylethyl)morpholin-3-yl]acetamide
1-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
8-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(oxolan-2-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]thiophene-2-carboxamide
3-(2-hydroxyphenyl)-N-[1-(1H-imidazol-1-yl)butan-2-yl]-1H-pyrazole-5-carboxamide
1-{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}-3-methylpiperidine
5-[(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]-2-methoxybenzoic acid
methyl (2S)-1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidine-2-carboxylate
N-(1-{1-[(2S)-2-acetamidopropanoyl]piperidin-4-yl}-2-(2-methylphenyl)ethyl)-N-methyl-2-(1H-pyrazol-1-yl)acetamide
7-[(4-fluorophenyl)methyl]-2-[2-(pyridin-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-(3-methoxypropyl)-1-[4-(methylsulfanyl)benzoyl]piperidine-3-carboxylic acid
(2S,4R)-4-(cyclooctylamino)-N-methyl-1-(2-methylpropyl)pyrrolidine-2-carboxamide
1-(3-fluorobenzoyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
4-[2-({4-[1-(furan-3-ylmethyl)piperidin-3-yl]-5-methylpyrimidin-2-yl}sulfanyl)ethyl]morpholine
8-[(3-chlorophenyl)methyl]-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
7-acetamido-N-[2-(1H-indol-3-yl)ethyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(5S,9aS,9bS)-5-(3,7-dimethyl-1H-indol-2-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3aR,5R,6S,7aS)-2-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]-octahydro-1H-isoindole-5,6-diol
N-{[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-methoxybenzamide
3-(2-chlorophenyl)-1-methyl-3-{2-oxo-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]ethyl}pyrrolidine-2,5-dione
(3R,4R)-1-(3-chlorobenzoyl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
ethyl 4-[4-(4-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
5-[3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carbonyl]quinoxaline
1-{3-[(2-fluorophenyl)methoxy]azetidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
(1S,5R)-3-(4-aminopyrimidin-2-yl)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-benzyl-N-(1,3-thiazol-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-{[7-chloro-2-(2,3-dimethoxyphenyl)quinolin-3-yl]methyl}cyclopropanamine
4-[2-(1-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethyl]morpholine
2,6-dimethoxy-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]pyrimidine-4-carboxamide