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(5S,9aS,9bS)-5-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
N-tert-butyl-7-(pyridine-2-amido)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-benzyl-7-chloro-N-(2-hydroxyethyl)-3,5-dimethyl-1-benzofuran-2-carboxamide
3-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-1-ethyl-4,6-dimethyl-1,2-dihydropyridin-2-one
4-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)-1,4-oxazepan-6-ol
1-ethyl-5-oxo-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidine-3-carboxamide
2-{[(3S,5S)-5-[4-(adamantan-2-yl)piperazine-1-carbonyl]-1-[(2,5-dimethylphenyl)methyl]pyrrolidin-3-yl]sulfanyl}-4-methylpyrimidine
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-methylpyridine
[1-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
(4aS,8aR)-6-[(2-ethylpyrimidin-4-yl)methyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1-({5-[(2,3-difluoro-4-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
2-[4-(thiomorpholin-4-yl)piperidin-1-yl]pyridine-3-carboxamide
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]pyridine-2-carbonitrile
(3R,4R)-4-ethyl-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}piperidine-3,4-diol
3-{[3-(3-benzoylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}-5-chloropyridine
(2S,4R)-1-(2,2-dimethylpropanoyl)-N-ethyl-4-[2-(thiophen-3-yl)acetamido]pyrrolidine-2-carboxamide
3-{[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
N-[2-(dimethylsulfamoyl)ethyl]-2-(2H-indazol-2-yl)acetamide
(4aR,8aR)-2-(2-hydroxypyridine-3-carbonyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
methyl[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl](oxolan-3-ylmethyl)amine
2-fluoro-6-hydroxy-N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]benzamide
N-(2-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(naphthalen-2-yl)acetamide
4-[4-(2-cyclopentyl-2-phenylacetyl)piperazin-1-yl]-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-N-(propan-2-yl)pyridine-4-carboxamide
1-(2-{[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}pyrimidin-4-yl)piperidin-3-ol
3-[5-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
5-[3-(4-chlorophenyl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-ethyl-N-(2-oxo-2-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}ethyl)cyclohexane-1-carboxamide
1-[3-(2-methoxyphenyl)phenyl]-3-[3-(oxolan-3-yl)propyl]urea
3-(4-chloro-2-methylbenzoyl)-1-(cyclopent-1-ene-1-carbonyl)piperidine
(4aR,7aS)-1-cyclopropanecarbonyl-4-[(1-ethyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-3-propoxypiperidine
4-(1,3-benzothiazol-2-yl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
1-{4-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
2-{4-[(2,5-dimethoxyphenyl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
4-{1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}thiomorpholine
1-cyclopentyl-3-(2-methylphenyl)-3-{2-[4-(morpholine-4-carbonyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
4-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-N,N,5,6-tetramethylpyrimidin-2-amine
(9aS)-2-(3-fluoro-2-methoxybenzoyl)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
5-[({4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)methyl]-N-methylfuran-2-carboxamide
ethyl 2-({[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]carbamoyl}amino)acetate
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)[(4-methyl-1H-imidazol-2-yl)methyl](oxolan-2-ylmethyl)amine
(4aS,7aR)-1-(2,4-dimethylbenzoyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
7-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1-oxa-7-azaspiro[3.5]nonane
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[2-(pyridin-3-yl)piperidin-1-yl]ethan-1-one