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methyl 3-(cyclobutylmethoxy)-5-(3-hydroxypyrrolidine-1-carbonyl)benzoate
N-(2,5-dimethoxyphenyl)-3-(2-methoxybenzoyl)piperidine-1-carboxamide
1-(propan-2-yl)-2-(1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,2,3-triazol-4-yl)-1H-1,3-benzodiazole
2-benzamido-N-methyl-7-oxo-N-(propan-2-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-(2-{8-[2-(dimethylamino)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-[2-(1H-indol-1-yl)ethyl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
ethyl 1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N-({8-[(3-chlorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
N-ethyl-2-(4-methoxyphenoxymethyl)-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
1-[1'-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
(3aR,6aS)-2-ethyl-1-oxo-5-(prop-2-ene-1-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-(thiophen-2-ylmethyl)-1H-pyrazole-4-carboxamide
(1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
[(5-methylthiophen-2-yl)methyl]({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})(pyridin-4-ylmethyl)amine
1-methyl-7-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazolo[1,5-a]imidazole
5-[5-(ethoxymethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-(piperidine-3-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N,3,6-trimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-{[1-butyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,1-dimethyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-(2-{7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
ethyl 5-[(3,5-difluorophenyl)methyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(5-{[ethyl(oxolan-2-ylmethyl)amino]methyl}furan-2-yl)methanol
N-(1-{7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
methyl 5-{[1,2,3,4]tetrazolo[1,5-a]pyridine-5-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-[(1S,2R)-2-aminocyclobutyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-N-(1,3-thiazol-2-yl)propanamide
methyl 3-({2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazol-4-yl}formamido)propanoate
ethyl 4-[(2-chlorophenyl)methyl]-1-[3-(morpholin-4-yl)propanoyl]piperidine-4-carboxylate
1-cyclohexanecarbonyl-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(cyclopropylmethyl)piperidine-3-carboxylic acid
3-[(2R,3R,6R)-5-(3-chlorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
5-(2-chlorophenyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]furan-2-carboxamide
methyl 3-(furan-2-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{2-[4-(3-chloro-4-fluorophenyl)-1H-1,2,3-triazol-1-yl]ethyl}aniline
3-ethoxy-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]propan-1-one
1-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-4-(4-chlorophenyl)butan-1-one
5-(3,5-dichloro-4-methylbenzoyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
9-methoxy-N-(3-methylbutyl)-7-oxo-3-(2-phenylpropyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(4aS,8aR)-2-{3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-decahydroisoquinoline
1,6-dimethyl-4-oxo-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-1,4-dihydroquinoline-3-carboxamide
N-(4-fluorophenyl)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine-2-carboxamide
3-cyclopropyl-5-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1H-1,2,4-triazole
N-[(1-hydroxycyclohexyl)methyl]-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carboxamide
1-ethyl-3,5-dimethyl-N-{[5-(4-methylphenyl)-1,2-oxazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-methyl-2-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}-1H-1,3-benzodiazole
N-[4-(furan-2-yl)butan-2-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[(2R,3R)-1'-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
2-{[1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-yl]amino}-1-(pyrrolidin-1-yl)ethan-1-one