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1-[(3-fluorophenyl)methyl]-4-{1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
1-ethyl-5-(4-methylpiperidin-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2-{5-[(2-methylpiperidin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridine
N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)-2-(pyridin-4-yl)acetamide
2-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
1-methyl-3-{4-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]piperidine-1-carbonyl}-1,4-dihydroquinolin-4-one
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-phenylpropyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-(4-{2-methyl-3-[(pyridin-2-ylmethyl)amino]benzoyl}morpholin-3-yl)acetic acid
1-[(4-chlorophenyl)methyl]-N-(oxan-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(1-carbamoylcycloheptyl)-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
3-[(2-fluorophenyl)methyl]-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidine-3-carboxylic acid
methyl (2R,4S)-4-hydroxy-1-[3-(thiophen-2-yl)propanoyl]piperidine-2-carboxylate
4-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenol
N-[(2R,3R)-2-methoxy-1'-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
5-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carbonyl}pyrrolidin-2-one
1-(cyclopropylmethyl)-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylsulfanyl)acetamide
1-(4-benzylpiperazin-1-yl)-3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]propan-1-one
N-{1-[(5,6,7-trimethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidin-3-yl}acetamide
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2-(morpholin-3-yl)acetamide
4-tert-butyl-2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenol
N-[2-(4-methoxyphenyl)ethyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)ethan-1-one
1-[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propan-1-one
2-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperidin-3-ol
2-butyl-5-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole
5-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(4aS,7aR)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-methoxyethyl)-1-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
3-chloro-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
4-(2-fluorophenoxy)-1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
4-[2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzenesulfonyl]-2-(trifluoromethyl)morpholine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
N,2-dimethyl-2-({1-[1-(2-phenylethyl)piperidin-4-yl]piperidin-3-yl}formamido)propanamide
5-(3,4-dimethoxyphenyl)-N-propylfuran-2-carboxamide
1-(4-chlorophenyl)-N-(3,4-dihydro-2H-1-benzopyran-3-yl)piperidin-4-amine
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-1-cyclopentylpiperidine-3-carboxamide
3-[({1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-yl}oxy)methyl]pyridine
(4aR,7aS)-1-butyl-4-(2,5-difluorobenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-({cyclopropyl[(3-methylthiophen-2-yl)methyl]amino}methyl)-5-(hydroxymethyl)-2-methylpyridin-3-ol
3-{1-[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}pyridine
N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-(1H-pyrazol-1-ylmethyl)-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-oxazepane
2-hydroxy-1-{4-[methyl(thiophen-2-ylmethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one