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3-(1,3-benzoxazol-2-ylmethyl)-8-methoxy-3,4-dihydroquinazolin-4-one
1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
3-[1-(1-methyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)piperidin-3-yl]benzoic acid
4-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)piperidine-4-carboxamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3,3,3-trifluoropropyl)piperidine
2-butyl-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-4-(dimethylamino)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-yl]propanoic acid
5-(4-methanesulfonylphenyl)pyridin-3-amine
4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2-(2-methoxyethyl)morpholine
1-(difluoromethyl)-N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-1H-pyrazole-5-carboxamide
6-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2,4-dimethylpyridine-3-carbonitrile
2-(3-methoxyphenoxymethyl)-N-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-1,3-oxazole-4-carboxamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-(morpholin-4-ylmethyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
3-[(2R,3R,6R)-5-(6-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
3-(oxolan-3-yl)-5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,2,4-oxadiazole
3-(but-2-yn-1-yl)-5-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[2-(methylsulfanyl)pyridine-3-carbonyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
1-(oxolan-3-ylmethyl)-4-(2-phenoxyethyl)piperazine
1-(2-phenylethyl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-2-one
1-{5-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]thiophen-2-yl}ethan-1-one
N'-(2,4-dimethylphenyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]ethanediamide
2-{2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
4-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2,6-dimethylpyrimidine
N-cyclopropyl-3-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]propanamide
3-(2-methoxyphenyl)-1-methyl-3-{2-oxo-2-[3-(pyridine-3-carbonyl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[2-(1H-pyrazol-1-yl)phenyl]piperidine-1-carboxamide
4-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
3-({[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
N3-methyl-N3-[(4-phenoxyphenyl)methyl]piperidine-1,3-dicarboxamide
methyl 3-{[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylformamido]methyl}-5-(1,3-dimethyl-1H-pyrazole-5-amido)benzoate
4-(2-aminopyridine-4-carbonyl)-1-(2-chlorophenyl)-5-methylpiperazin-2-one
4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1-(2-methoxyphenyl)piperazin-2-one
5-{1-[2-(2,6-difluorophenyl)acetyl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)pent-4-enamide
N-[1-(1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
6-cyclopentyl-2-methoxy-3-{[(4-methylpyrimidin-2-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-(4-benzyl-1H-pyrazol-5-yl)-1-(2,3-dihydro-1H-inden-2-yl)piperidine
2-{methyl[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}acetamide
1-ethyl-4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazine
(3S,4S)-4-(pyridin-2-yl)-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)pyrrolidine-3-carboxylic acid
{[2-(butan-2-yloxy)phenyl]methyl}({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
2-cyclopropyl-5-{4-[(3-fluorophenyl)methyl]-3-oxopiperazine-1-carbonyl}-3,4-dihydropyrimidin-4-one
1-benzyl-3-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-3-methylurea
N-ethyl-2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-(2-hydroxyethyl)acetamide
2-(2-fluorophenoxymethyl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
methyl (2S,4S)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-[(3-ethoxy-4-hydroxyphenyl)methyl]pyrrolidine-2-carboxylate
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(8-{[4-(benzyloxy)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-1-methyl-1H-pyrazole-5-carboxamide