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3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-[1-(4-methylpentanoyl)piperidin-4-yl]imidazolidine-2,4-dione
4-({5-[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
6-methoxy-2-oxo-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-[5-(dimethylcarbamoyl)thiophen-2-yl]thiophene-2-carboxylic acid
1-(4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
2,8-dimethyl-3-[3-(pyridin-4-yl)azetidine-1-carbonyl]quinoline
3-(4-chlorobenzoyl)-1-[(2,4-dimethoxyphenyl)methyl]piperidine
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-3-(2-ethylphenoxy)azetidine
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
2-fluoro-N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indazole
9-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)benzamide
methyl 4-{[2-(hydroxymethyl)piperidine-1-carbonyl]amino}-3-methylbenzoate
(3R,4S)-4-cyclopropyl-1-[5-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-5-methylpyrazine-2-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-6-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
N-(1-benzylpiperidin-4-yl)-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(5-phenyl-4H-1,2,4-triazol-3-yl)ethan-1-one
1-(3-chlorophenyl)-4-(3-phenyl-1H-pyrazole-4-carbonyl)piperazin-2-one
ethyl 4-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
N-(1-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
5-methyl-1-(4-methylphenyl)-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperazin-2-one
N-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
3-(1-phenylpiperidin-4-yl)-3,4-dihydropteridin-4-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1H-imidazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[4-(4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperazin-1-yl]phenol
2-(1-benzofuran-2-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
methyl 1-[(3S,5S)-1-(2-ethylbutyl)-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[(prop-2-en-1-yl)amino]-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
N-(dicyclopropylmethyl)-3-[(4-methoxyphenyl)methyl]-1,2-oxazole-5-carboxamide
8-chloro-2-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-ylmethyl)quinolin-4-ol
7-(2-hydroxyethyl)-2-[2-(methylamino)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-2-(1,3-thiazol-2-yl)piperidine
N-[(8-{[4-(furan-2-yl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
N-(furan-2-ylmethyl)-4-[4-(thiomorpholin-4-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
ethyl 4-(cyclopropylmethyl)-1-(2,5-dimethoxybenzenesulfonyl)piperidine-4-carboxylate
(1R,5S,6S)-6-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(oxolan-2-yl)acetamide
(2E)-3-(4-fluorophenyl)-N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
1-(1H-imidazol-2-ylmethyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
3-({[(4-fluoro-2-methoxyphenyl)methyl]amino}methyl)-N,N-dimethylpyridin-2-amine