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methyl 2-(1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-N-methylformamido)acetate
1-cyclohexyl-N-methyl-4-oxo-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,4-dihydropyridine-3-carboxamide
(1S,5R)-1,3,3-trimethyl-6-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-6-azabicyclo[3.2.1]octane
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
2-[cyclopentyl(methyl)amino]-1-[3-(2-methylphenoxy)azetidin-1-yl]ethan-1-one
3-(2-chlorobenzoyl)-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)acetamide
(2S)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-oxopyrrolidine-2-carboxamide
2-(furan-2-yl)-5-{1-[1-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
N-(3-acetamido-4-methoxyphenyl)-3-(2-ethylphenoxy)azetidine-1-carboxamide
5-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
(3S,5R,9R)-11-(4-chlorobenzoyl)-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-[2-(methylsulfanyl)ethyl]-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
3-(1-methyl-1H-imidazol-2-yl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
3-({methyl[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino}methyl)benzoic acid
3-[(2,3-dimethoxyphenyl)methyl]-5-{1-[3-(dimethylamino)benzoyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
4-(4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)quinazoline
7-(1-ethyl-1H-pyrazole-4-carbonyl)-N,N-dimethyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{2-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxolane-2-carboxamide
2-(2H-indazol-2-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
ethyl 1-(cyclopropylmethyl)-5-[1-(pyridin-2-yl)piperidine-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{[5-(2-methoxy-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-methyl-1,2-oxazole
3-[benzyl(quinolin-3-ylmethyl)amino]-2-methylpropan-1-ol
(9aR)-2-methyl-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3R,4R)-3-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-4-ol
2-methanesulfonamido-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethan-1-one
4-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}thiomorpholine
3-{2-[1-(4-chloro-2-fluorobenzoyl)piperidin-2-yl]ethyl}phenol
methyl 3-{[5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-yl]amino}propanoate
(1S,5R)-6-(5-methyl-1,2-oxazole-3-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
5-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(4-methyl-1H-imidazole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(pyrimidin-2-yl)-1,4-diazepane
1-[benzyl(methyl)amino]-3-[2-methoxy-5-(morpholin-4-ylmethyl)phenoxy]propan-2-ol
3-chloro-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyridin-2-amine
4-(piperidine-1-carbonyl)-1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
3-chloro-4-{3-[1-(dimethylamino)ethyl]phenyl}benzoic acid
(1r,4r)-4-({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)cyclohexan-1-ol
3-(2H-1,3-benzodioxole-5-carbonyl)-N,N-dimethylpiperidine-1-sulfonamide
1-{7-[(1-methyl-1H-imidazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine-3-carbonitrile
3-cyclobutyl-4-[2-(2-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 2-({4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]phenyl}formamido)acetate
N-[(3-methyl-7-{2-[3-(trifluoromethyl)phenyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1,3-thiazole-5-carboxamide
3-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-ylmethyl]-N-(1-methyl-1H-pyrazol-5-yl)benzamide
2-(2,4-dimethoxyphenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
N-cyclopropyl-3-(5-sulfamoylthiophen-2-yl)benzamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-(9H-purin-6-yl)piperidin-4-amine
1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
N-({7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide