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3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
N,N-diethyl-1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxamide
1-methyl-3-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1,2-dihydroquinolin-2-one
6-[(3-fluorophenyl)methoxy]-4-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-1-(2-methylpropyl)-1,4-diazepan-2-one
6-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]pyridine-3-carboxamide
5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1H-indole
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-2-(2-oxoazepan-1-yl)acetamide
7-(3,4-dimethoxyphenyl)-9-methoxy-4-[(3-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-(3,4-dihydronaphthalen-2-yl)-4-[(4-methyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
9-(2,5-dimethylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-({2-[(4-chlorophenyl)methyl]-1,3-benzoxazol-5-yl}formamido)acetamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-ethyl-2-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1H-indole
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-indole-2-carboxamide
2-{2-oxo-2-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethyl}-3-phenylcyclopent-2-en-1-one
7-[(2-fluorophenyl)methyl]-2-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,7-diazaspiro[4.5]decane
{1-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]pyrrolidin-3-yl}methanamine
3-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyridazine-3-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
3-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-4-methylbenzene-1-sulfonamide
N-methyl-2-(2-oxo-1,2-dihydropyridin-1-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(2-phenoxyethyl)amine
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-(pyrrolidin-1-yl)butanamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-methyl-N-(oxolan-3-yl)-1,2-oxazole-3-carboxamide
N-{[2-(benzyloxy)phenyl]methyl}-2-ethylpyrimidine-5-carboxamide
5-[1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)pyrrolidin-2-yl]-N-methylthiophene-2-carboxamide
N-benzyl-1-cyclopropyl-N-[(6-methylpyridin-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-(oxolan-2-ylmethyl)-3-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1,2-oxazole-5-carboxamide
5-ethyl-6-methyl-N4-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidine-2,4-diamine
9-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-(dimethylamino)-2-(3-methylphenyl)-1-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}ethan-1-one
{4-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
[(3R,5S)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
3-cyclohexyl-N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(2-chlorophenyl)methyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
6-methyl-2-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)pyridin-3-ol
N-{[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
7-(1,3-benzothiazol-2-yl)-4-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(butan-2-yl)-5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
6-methyl-2-oxo-5-({2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridine-3-carbonitrile
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
6-[(diethylamino)methyl]-N-[(2R)-2-hydroxypropyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-cyclohexyl-5-{1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}pyrimidine
N-[(2,6-difluoro-3-methylphenyl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
1-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-N-methylpiperidine-2-carboxamide
2-{[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]methyl}-6-fluoroquinolin-4-ol
(2R)-2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidine