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(4aR,7aS)-1-(2-{methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2-hydroxyphenyl)ethan-1-one
3-(hydroxymethyl)-N-[4-(4-methoxyphenyl)phenyl]piperidine-1-carboxamide
1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-(2-ethoxyphenyl)ethan-1-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-4-methoxy-N-(2-methoxyethyl)-3-methylbenzamide
2-(2-methyl-1,3-thiazol-4-yl)-N-(3-{[(2-methylphenyl)methyl]sulfanyl}propyl)acetamide
2-[benzyl(methyl)amino]-N-[2-(pyridin-3-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-(1-phenylpiperidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
2-{[methyl({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}pyridine-3-carboxylic acid
5-[1-(2-phenylbenzoyl)pyrrolidin-2-yl]thiophene-2-carboxamide
3-fluoro-4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
5-[3-(2-methylphenoxymethyl)piperidine-1-carbonyl]isoquinoline
ethyl 4-(cyclopropylmethyl)-1-{[4-(methoxycarbonyl)phenyl]methyl}piperidine-4-carboxylate
4-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}quinoline
N-({1-[(2,4,5-trimethylphenyl)methyl]pyrrolidin-3-yl}methyl)pyrimidine-5-carboxamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(pyrimidin-2-yl)-1,4-diazepan-5-one
N,2-dimethyl-N-[2-(methylsulfanyl)ethyl]thieno[3,2-d]pyrimidin-4-amine
2-(adamantan-1-yl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
(3S,4S)-4-propyl-1-(1,3-thiazol-2-ylmethyl)pyrrolidine-3-carboxylic acid
methyl 2-{2-[(2S,4R,6R)-6-tert-butyl-4-acetamidooxan-2-yl]phenoxy}acetate
N-(4-{1-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-1H-imidazol-2-yl}phenyl)acetamide
(3S,4R)-1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4-methylpiperidine-3,4-diol
2-(2H-1,3-benzodioxol-5-yl)-5-(1H-indol-2-ylmethyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
3-chloro-2-[4-(1H-pyrazol-5-yl)phenyl]pyridine
4-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2,2,3-trimethylbut-3-en-1-one
5-(3-fluorophenoxymethyl)-N-[1-(pyridin-2-yl)propyl]-1H-pyrazole-3-carboxamide
N-(2-methyl-4-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenyl)acetamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]propan-1-one
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl){[2-(trifluoromethyl)phenyl]methyl}amine
3-{4-[5-(1-benzofuran-2-yl)-1,2,4-triazin-3-yl]piperazin-1-yl}-1λ6-thiolane-1,1-dione
4-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoline
8-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(3-propoxypiperidin-1-yl)pyridine-3-carboxamide
5-benzenesulfonamido-1-ethyl-N,2-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
2-methyl-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-(2-methylphenyl)piperazine
2-(1-methyl-1H-pyrazole-5-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
3-(2-methoxyethyl)-1-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-3-(1,3-thiazol-2-ylmethyl)urea
ethyl 2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
4-{5-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}-1H-indole
N-(2-hydroxyethyl)-5-[6-(piperidin-1-yl)pyrimidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-benzyl-4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidine-1-carboxamide
dimethyl[1-(3-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenyl)ethyl]amine
2-[1-(propan-2-yl)-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazin-2-yl]ethan-1-ol
(1R,5S,6R)-3-{[2-(5-methylfuran-2-yl)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}oxane-2-carboxamide
3-(cyclopropylsulfamoyl)-N-(oxan-4-yl)benzamide
1-{[2-hydroxy-5-(pyrazin-2-yl)phenyl]methyl}piperidin-3-ol