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7-chloro-4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-({4-[3-(pyrrolidin-1-yl)pyrazin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-4-(5-methylfuran-2-yl)benzamide
1-(furan-3-ylmethyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
11-{[(2-fluorophenyl)methyl]amino}-4-(pyridin-4-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(4-fluorophenyl)methyl]-N-[2-(6-methylpyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
1-[(5-ethylpyridin-2-yl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
3-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
[1-(1H-imidazol-1-yl)propan-2-yl](4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)amine
2-ethyl-4-phenyl-9-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,5S,8S)-3-[(6-ethoxypyridin-3-yl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
1-(3-methyloxetane-3-carbonyl)-3-propylpiperidine-3-carboxylic acid
3-(methoxymethyl)-1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidine
3-(1-methanesulfonylpiperidin-4-yl)-1-[3-(pyridin-3-yl)phenyl]urea
N-[2-(2-methylphenyl)-1,3-benzoxazol-6-yl]-6-oxo-1,6-dihydropyridine-2-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
N-methyl-1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]pyrrolidine-3-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-cycloheptyl-N-methyl-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
3-(5-methyl-1H-pyrazol-1-yl)-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}propanamide
2-[4-(1-methoxyethyl)phenyl]-4-(piperidine-1-carbonyl)pyridine
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)(pyridin-2-ylmethyl)amine
ethyl 3-{[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazol-3-yl]formamido}-4-methylpentanoate
3-[({3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}amino)methyl]pyrrolidin-3-ol
(3S,4S)-1-[(3-ethoxy-4-hydroxyphenyl)methyl]-4-(4-fluorophenyl)piperidin-3-ol
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,8-dimethylimidazo[1,2-a]pyridine-2-carboxamide
3-[benzyl({[1-(propan-2-yl)piperidin-4-yl]methyl})amino]-2-methylpropan-1-ol
3-(azocan-1-yl)-N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropylpropanamide
N-[4-fluoro-3-(2-methylpropanamido)phenyl]-4-[(methylsulfanyl)methyl]piperidine-1-carboxamide
3-(5-chloro-2-methoxypyridin-4-yl)-6-(pyrrolidin-1-yl)pyridazine
methyl 5-(pyrimidin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-(1H-indol-3-yl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-cyclopropyl-4-(3-fluorophenyl)-N-({4-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)benzamide
N-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-N-methylthian-4-amine
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(5-oxopyrrolidin-2-yl)acetamide
2-{4-[(4-ethoxyphenyl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(1-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanamine
5-methyl-N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
5-[1-(4-fluoro-3-methylbenzoyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
1-phenyl-4-[1-(1-phenylpiperidin-4-yl)piperidin-3-yl]piperazine
3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-8-methyl-3,4-dihydroquinazolin-4-one
N-(1-{7-[(2-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylbenzamide
N-ethyl-2,5-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)furan-3-carboxamide
N-{[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-methylbutanamide
4-benzyl-3-[2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-(1-ethyl-5-oxopyrrolidin-3-yl)-2,6-dihydroxybenzamide