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(4aR,7aS)-N,N-dimethyl-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-[(1R,2R,3S,4S)-3-aminobicyclo[2.2.1]heptane-2-carbonyl]-1-(2-methoxyphenyl)piperazin-2-one
2-(oxolan-3-yl)-1H-1,3-benzodiazole-6-carboxylic acid
1-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2,2-dimethylpropan-1-one
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1H-pyrrole-3-carbonyl)piperidin-3-yl]propanamide
2-{5-[1-(1,3-thiazol-4-ylmethyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
N,N,5-trimethyl-2-[4-(3-methylpyridin-4-yl)piperazin-1-yl]pyrimidin-4-amine
2,2-dimethyl-N-(3-{[methyl({2-[(4-methylphenyl)sulfanyl]ethyl})amino]methyl}pyridin-2-yl)propanamide
3-(2-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
4-(morpholin-4-yl)-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-2-amine
3-(5-fluoro-2-methoxybenzoyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-(1-methylpiperidin-4-yl)-N'-[2-(methylsulfanyl)phenyl]butanediamide
(2R)-2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
5-chloro-4,6-dimethyl-2-oxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2-dihydropyridine-3-carboxamide
3-{4-[2-(3-ethoxyphenoxy)ethyl]piperazin-1-yl}pyrazine-2-carbonitrile
1-(cyclohexylmethyl)-5-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]piperidin-2-one
2-chloro-N-{[1-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-3-yl]methyl}benzamide
4-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-phenylpiperazin-2-one
3-methyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-5-propyl-1-benzofuran-2-carboxamide
N-[3-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)-4-fluorophenyl]propanamide
3-[2-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-2-oxoethyl]-2,3-dihydro-1H-isoindol-1-one
2-(benzyloxy)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
1-(cyclopropylmethyl)-5-[2-(methylamino)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(1S,3R)-3-amino-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]cyclopentane-1-carboxamide
6-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-5-{1-[(2E)-4-methylpent-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
2-(2-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
3-chloro-N-(3-hydroxy-3-methylbutyl)-5-methoxy-N-methylbenzamide
1-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
N-(1H-imidazol-2-ylmethyl)-1-(2-methoxyethyl)-N-methyl-6-oxopiperidine-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-(morpholine-4-carbonyl)pyridin-2-amine
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
1-[(3-methylpyridin-2-yl)methyl]-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
N-[(3S,4R)-1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-propylpyrrolidin-3-yl]acetamide
2-methyl-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(furan-2-ylmethyl)-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}piperidine
(3S,4S)-1-(propan-2-yl)-4-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]pyrrolidin-3-ol
{2-ethoxy-5-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}amino)methyl]phenyl}methanol
4-{5-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
1-(4-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}phenyl)imidazolidin-2-one
N-(2-hydroxyethyl)-2-(morpholin-4-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(pyridin-3-yl)acetamide
1-{3-[(1,4-dithiepan-6-yl)amino]propyl}piperidin-3-ol
N-(1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
methyl 3-[(2,4-difluorophenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[(1-acetylpiperidin-4-yl)oxy]-N-(1H-indol-2-ylmethyl)-5-methoxybenzamide
1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
3-{1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
1-{2,7-diazaspiro[4.5]decan-7-yl}-2-(pyridin-3-yloxy)ethan-1-one
4-{pyrazolo[1,5-a]pyrimidin-3-yl}-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine