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1-{2-oxo-2-[3-(2-phenylethyl)piperidin-1-yl]ethyl}pyrrolidin-2-one
2-cyclopentyl-N-{[(2S,4S)-4-fluoro-1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]pyrrolidin-2-yl]methyl}acetamide
1-[3-oxo-3-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propyl]pyrrolidin-2-one
4-{2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-ylmethyl]-1H-pyrrol-1-yl}benzonitrile
2-(methylsulfanyl)-N-[1-(pyridin-3-yl)propan-2-yl]pyridine-3-carboxamide
2-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
2-[3-(methylsulfanyl)propyl]-2,8-diazaspiro[4.5]decane
7-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-2-oxa-7-azaspiro[4.5]decane
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-propylacetamide
(1R,5R)-6-[(5-chlorothiophen-2-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-3-methoxy-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-4-amine
4-[(2S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
3-(3-hydroxy-3-methylbutyl)-N-(1-phenylpiperidin-4-yl)benzamide
4-(2-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-yl}ethyl)morpholine
3-[(4-fluorophenyl)methyl]-5-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
7-[3-(propan-2-yloxy)phenyl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
N-(3,5-dimethoxyphenyl)-3-{1-[3-(1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}propanamide
3-(2-methylpropyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1,2-oxazole-5-carboxamide
3-methyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
1-[2-(furan-2-yl)pyrrolidin-1-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
(2R,6S)-4-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}-2,6-dimethylmorpholine
5-(2-chlorophenyl)-N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]furan-2-carboxamide
7-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
4-[(2,5-dimethoxyphenyl)methyl]-9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-methylpiperazin-1-yl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-6-(thiophen-3-yl)pyridine-3-carboxamide
[(4-fluorophenyl)methyl]({[5-methyl-1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})(pyridin-4-ylmethyl)amine
5-(4-chloro-2-methoxyphenoxymethyl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
1-[(4-fluoro-3-methylphenyl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
2-methyl-4-(2-methylphenyl)-1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
N-(2-methanesulfonamidoethyl)-4-(1H-pyrazol-3-yl)benzamide
N-[(1-butyl-1H-1,2,4-triazol-5-yl)methyl]-4-fluoro-3-methylbenzene-1-sulfonamide
4-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholine
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
4-fluoro-3-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzene-1-sulfonamide
N-[(2-methoxyphenyl)methyl]-2-oxo-N-(prop-2-en-1-yl)-2H-chromene-3-carboxamide
6-methyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-phenylpyrimidin-4-amine
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
1,2-dimethyl-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
(3aR,6aS)-5-(2,1-benzoxazole-3-carbonyl)-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[(2,3-dimethoxyphenyl)methyl]-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-methyl-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,2-oxazole-3-carboxamide
2-(2-hydroxyphenyl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
(4aR,7aS)-1-ethyl-4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-1-(2,6-difluorobenzoyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-3-[2-(3-methylpiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
4-[2-(1,2-benzoxazol-3-yl)acetyl]-1-(1H-indazol-6-yl)piperazin-2-one
N-(2-hydroxyethyl)-1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-3-yl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-({[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amino}methyl)-2,6-dimethylphenyl acetate