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N-[2-(2-chlorophenyl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
7-methyl-3-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]-N-methylpyrazin-2-amine
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
N-cyclopentyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)pent-4-enamide
2,3,5,6-tetramethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]benzamide
1-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-(3,4-dichlorophenyl)ethan-1-one
N-[2-(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)ethyl]acetamide
4-{1-[6-(4-methylpiperazin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
7-(pyridin-3-yl)-4-(pyrimidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
pyridin-2-yl({1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl})methanol
4-(1-hydroxy-3-methylbutan-2-yl)-11-methyl-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl][2-(oxan-4-yl)ethyl]amine
2-[(4-methoxyphenyl)methyl]-4-{4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N,1-dimethyl-N-[(4-{[1-(pyridine-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperidin-4-amine
1-[5-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)thiophen-2-yl]ethan-1-one
3-{1-[2-(carbamoylamino)acetyl]piperidin-3-yl}-N-[(3,4-difluorophenyl)methyl]propanamide
9-(cyclopropylmethyl)-4-(5,6-dimethylpyrimidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[1-(3-methylbutyl)-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl]ethan-1-ol
4-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]benzoic acid
1-[4-(furan-2-carbonyl)piperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-5-(1,3-thiazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1-{5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}piperidin-2-yl)methanol
N-cyclopropyl-2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
(2R,4S)-1-(4-tert-butylbenzoyl)-4-hydroxypiperidine-2-carboxylic acid
3-(6-chloropyridin-3-yl)-1-[(3-methoxyphenyl)methyl]-1-(3-methoxypropyl)urea
2-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(1-benzoxepine-4-carbonyl)-N-cyclopropylpiperazine-2-carboxamide
2-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]-N-(propan-2-yl)benzamide
4-benzyl-1-methyl-3-[1-(prop-2-ene-1-sulfonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(morpholin-4-yl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
(3S,4S)-1-(1H-imidazol-2-ylmethyl)-4-(3-methoxyphenyl)piperidin-3-ol
7-[(4-fluorophenyl)methyl]-2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decane
5,6,7-trimethoxy-N,N-dimethyl-3-({[1-(naphthalen-1-yl)ethyl]amino}methyl)quinolin-2-amine
1-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-3-yl}-2-phenylethan-1-one
1-[7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
methyl 4-{4-[2-(2-fluorophenyl)-1-[N-methyl-3-(methylsulfanyl)propanamido]ethyl]piperidin-1-yl}-4-oxobutanoate
2-(4-chlorophenyl)-4-(4-propylpyrimidine-5-carbonyl)morpholine
3-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]-1-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}urea
[2-(1-phenyl-1H-pyrazol-4-yl)ethyl](4,4,4-trifluorobutan-2-yl)amine
[(3R,4S)-1-{[2-(difluoromethoxy)phenyl]methyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(cyclopropylmethyl)-3-hydroxy-3-[({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)methyl]piperidin-2-one
1-[4-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)phenyl]-1H-1,2,4-triazole
1-(furan-2-ylmethyl)-1-methyl-3-{5-[2-(morpholin-4-yl)ethyl]-1,3,4-thiadiazol-2-yl}urea
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-methyl-1,2-dihydroquinolin-2-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(piperidin-3-yl)benzamide
3-chloro-7-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrazolo[4,3-c]pyridine