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2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[1-(4-methoxyphenyl)ethyl]-N-methylacetamide
N-(adamantan-2-ylmethyl)-6-{[benzyl(methyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrazine
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2-(pyridin-2-yl)acetamide
4-(1H-imidazol-2-yl)-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
4-cyclohexyl-3-{[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-4H-1,2,4-triazole
(2S)-3-phenyl-2-{[3-(1H-pyrazol-1-ylmethyl)phenyl]formamido}propanamide
3-(2-cyclohexylethyl)-4-methoxybenzamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-diphenylacetamide
N-[(2R,3R)-1'-[(3,5-dimethoxyphenyl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
3-(2-amino-1,3-thiazol-4-yl)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}propan-1-one
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butan-1-one
1-[2-(4-methoxyphenyl)ethyl]-8-[(2-methylphenyl)methyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[1-(diethylsulfamoyl)piperidin-3-yl]benzoic acid
2-methoxy-3-[3-(2-methoxyphenoxy)azetidin-1-yl]pyrazine
6-[1-(4-chlorophenyl)cyclobutanecarbonyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,1-dimethylazepane-2-carboxamide
3-{8-chloro-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl}pyridine
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(2-phenyl-1,3-thiazol-4-yl)methyl]amine
2-[benzyl({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
6-[(diethylamino)methyl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(2-fluorophenoxymethyl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)piperidine-1-carboxamide
2-(4-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
1-[2-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-[1-(2-methylpyridine-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
4-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]piperidin-1-yl}-N-(1-phenylethyl)benzamide
5-amino-N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-4-phenyl-1H-pyrazole-3-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
7-(2,3-dihydro-1H-inden-2-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-benzyl-N-ethyl-1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
N-benzyl-1-[2-(2,2-dimethylpropanamido)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carboxamide
3-(4-chlorophenyl)-N-methyl-3-phenyl-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
(4aS,8aR)-2-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-decahydroisoquinoline
4-(hydroxymethyl)-1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-ol
methyl N-(1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-1-oxopropan-2-yl)carbamate
2-(furan-2-yl)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-oxoacetamide
3-(2-methyl-1H-imidazol-1-yl)-1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}propan-1-one
8-[(2-methylphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{5-benzyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}pyrrolidin-3-amine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
4-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
2-(methylamino)-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]ethan-1-one
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine