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2-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-2,3-dihydro-1H-isoindole
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-1-(morpholin-4-yl)cyclohexane-1-carboxamide
N-benzyl-N-ethyl-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetamide
N-benzyl-2-ethyl-7-(2-methoxybenzamido)-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(1H-indol-4-ylmethyl)-5-methoxybenzamide
1-(4-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-one
(4aS,8aR)-1-(4-hydroxybutyl)-6-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[4-({3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]acetamide
5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-N-ethyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3,5-dimethyl-1-[(4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}phenyl)methyl]-1H-pyrazole
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-[cyclohexyl(methyl)amino]-3-(2-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
5-[4-(2-phenylethyl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyridine
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-(methylsulfanyl)ethan-1-one
1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-3-phenylpyrrolidin-3-ol
methyl 1-[7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carbonyl]piperidine-2-carboxylate
N-(2-phenylethyl)-1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(6-methylpyridin-2-yl)methyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(4aS,7aR)-1-(3-phenylpropyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-({[2-(azepan-1-yl)ethyl](ethyl)amino}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-(2-fluorophenyl)-4-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
2-methyl-5-(3-methylphenyl)-4-[1-(1-methylpiperidine-4-carbonyl)piperidin-3-yl]pyrimidine
N-butyl-4-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(2-methoxypyrimidine-5-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(2-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
1-{4-[3-({[(2-chloro-6-fluorophenyl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
3-[2-(azocan-1-yl)-2-oxoethyl]-4-[(3,5-dimethoxyphenyl)methyl]piperazin-2-one
[3-ethyl-1-({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-3-yl]methanol
1-(3-aminoazepan-1-yl)-4-(benzyloxy)butan-1-one
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxylic acid
1-methyl-3-[4-(thian-4-yl)piperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
3-({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
2-{4-[(4-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-2-(3-methoxyphenyl)acetic acid
1-benzyl-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
(4aR,7aS)-1-[2-(azonan-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-5,5-diphenylpiperidin-2-one
1-(2-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)piperidine
N-({4-hydroxy-1-[(5-methylthiophen-2-yl)sulfonyl]azepan-4-yl}methyl)-2-methoxyacetamide
2-(2-chlorophenoxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
2-{3-[2-(dimethylamino)-2-(4-fluorophenyl)acetamido]propanamido}acetic acid
4-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-4-oxobutane-1-sulfonamide
2-[4-({methyl[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenyl]-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
N-(2-{7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
N-{1-[3-(piperidin-4-ylmethyl)benzoyl]piperidin-4-yl}pyrimidin-2-amine
methyl (2S)-1-{3-[2-(2-fluorophenyl)acetyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}pyrrolidine-2-carboxylate
[(2-chloro-5-ethoxy-4-propoxyphenyl)methyl](methyl)[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amine