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6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-2,3-dimethylquinoxaline
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
4-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
N-[(2-{4-[5-(methoxymethyl)thiophene-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
N-{2-[(pyridin-3-yl)amino]ethyl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
[(4,6-dimethylpyridin-2-yl)methyl][(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
N4-(1-benzylpyrrolidin-3-yl)-5-ethylpyrimidine-2,4-diamine
5-methoxy-2-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}pyridin-4-ol
3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]urea
2-[2-(thiophen-2-yl)ethyl]-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
1-ethyl-2-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-1H-1,3-benzodiazole
N-(2-methoxyethyl)-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-(pyridin-3-ylmethyl)benzamide
dimethyl[(5-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}thiophen-3-yl)methyl]amine
1-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-methoxy-2-methylpropanamide
3-(5-{7-methylthieno[3,2-d]pyrimidin-4-yl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
4-(1H-1,3-benzodiazol-1-yl)-1-(1-benzofuran-2-ylmethyl)piperidine-4-carboxylic acid
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-ethyl-1-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)piperidine
1-[1-(3-methylbenzoyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-[(5-methylfuran-2-yl)methyl]acetamide
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)propanamide
5-(2,6-dimethylphenoxymethyl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
5-acetyl-N-methyl-N-[1-(pyridin-3-yl)pentyl]thiophene-3-carboxamide
1-(3-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}phenyl)imidazolidin-2-one
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
5-(4-chloro-3-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2,6-dimethoxy-4-[1-(1-phenylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenol
2-[N-methyl-1-(3,5,7-trimethyl-1H-indol-2-yl)formamido]-2-(pyridin-3-yl)acetic acid
1-(azepan-1-yl)-3-[2-methoxy-4-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
4-[(2,3-dimethoxyphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
4-{2-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}morpholine
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)piperidine-1-carboxamide
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]morpholine-4-carboxamide
3-[4-(dimethylamino)phenyl]-N-(2-oxoazepan-3-yl)propanamide
3-[2-(pyridin-3-yl)-1,3-benzoxazol-5-yl]propanamide
2-methyl-N-[2-(pyrazin-2-yl)ethyl]thieno[3,2-d]pyrimidin-4-amine
2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-N-[(5-methylfuran-2-yl)methyl]quinazolin-4-amine
N-[4-(4-{[2-(2-methoxyphenyl)ethyl]amino}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
2-[4-(cyclopropylmethyl)-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
2-(1H-imidazol-2-ylmethyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(4-chloro-2-fluorophenyl)-1-ethyl-1-(oxan-4-ylmethyl)urea
2-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)acetic acid
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-1,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
3-{3-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-3-oxopropyl}oxolan-2-one
2-{[(1-methyl-1H-imidazol-2-yl)methyl](pyridin-3-ylmethyl)amino}butan-1-ol
4-(4-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
3-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
N-cyclopropyl-N-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2-methylpropanamide
methyl 4-[4-({4-[(4-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}methyl)-5-methyl-1,3-oxazol-2-yl]benzoate