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ethyl 1-[7-oxo-2-(thiophene-3-amido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carbonyl]piperidine-3-carboxylate
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2-methylpropyl)-1H-pyrazole-3-carboxamide
(1S,6R)-9-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-3,9-diazabicyclo[4.2.1]nonane
3-(2-ethyl-3-methyl-1-benzofuran-7-yl)-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
N-[(3-fluorophenyl)methyl]-9-methoxy-7-oxo-3-(pyridin-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
3-methoxy-5-methyl-N-[2-(piperidin-1-yl)ethyl]thiophene-2-carboxamide
N3-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-{1-[2-(1H-1,3-benzodiazol-1-yl)propyl]piperidin-4-yl}ethan-1-ol
2-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]quinoline
1-(3,4-dimethylphenyl)-3-methyl-3-[(4-methyl-1H-imidazol-2-yl)methyl]urea
2-[2-(1H-indol-3-yl)ethyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
5-{1-[3-(1H-pyrrol-1-yl)benzoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]acetamide
6-{1-[2-(trifluoromethyl)phenyl]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-cyano-N-(4-fluoro-3-methylphenyl)piperidine-1-carboxamide
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
(4aS,7aR)-1-(morpholine-4-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
dimethyl({2-[4-(1-phenyl-1H-pyrazole-4-carbonyl)morpholin-2-yl]ethyl})amine
4-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidin-2-amine
2-[4-(5-acetyl-4-methylpyrimidin-2-yl)piperazin-1-yl]pyridine-3-carbonitrile
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}propanamide
5-(2,5-dimethylfuran-3-carbonyl)-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1,3,6-trimethyl-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[4-(1-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]piperidine
N-methyl-3-[4-(3-methylphenyl)piperazin-1-yl]-N-[1-(1,2-oxazol-3-yl)ethyl]propanamide
1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
1-ethyl-8-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-4-(trifluoromethyl)pyridin-2-amine
3-(3-hydroxypropyl)-4-[2-(propan-2-yl)phenyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyridin-2-amine
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-(2-hydroxybutyl)pyrimidine-5-carboxamide
N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[(2R,3R)-2-methoxy-1'-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
2-{1-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]pyrrolidin-3-yl}benzoic acid
2-methoxy-5-[(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]pyridine
1-{2-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]morpholin-4-yl}ethan-1-one
4-{4-[1-(4-methoxy-2-methylphenyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-2,4-dimethoxybenzamide
1-(4-chloro-3-methylphenyl)-3-ethyl-3-(4-hydroxybutyl)urea
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
N-[1-(2,8-dimethylquinoline-4-carbonyl)piperidin-4-yl]acetamide
2-methoxy-1-[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-{3-[2-(2-hydroxyphenoxy)acetamido]phenyl}-2-methoxybenzamide
8-(3-fluoropyridine-4-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide