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N-[(2,3-difluorophenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-amine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
3-(5-{[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
2-[(1S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
(1S,5R)-6-benzyl-3-(3-hydroxypyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S)-2-amino-1-(4-{[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)propan-1-one
2-(cyclopent-1-ene-1-carbonyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-cyclopentyl-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
[(3R,5R)-1-(2-ethylpyridine-4-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
3-({4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazin-1-yl}methyl)phenol
N-(2-chloro-6-methylphenyl)-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
3-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-2-yl]pyridine
1-[(4-chlorophenyl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-(5-fluoro-2-methylbenzenesulfonyl)-3-(2-methoxybenzoyl)piperidine
8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-benzyl-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-methyl-2-(3-methylthiophen-2-yl)-4-{[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1,3-oxazole
(3-ethyl-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-yl)methanol
1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
3-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-[2-(propan-2-yloxy)phenyl]urea
5-(2-methoxyacetamido)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
(2S,4S)-4-amino-N-[2-(4-ethoxyphenyl)propan-2-yl]-1-methylpyrrolidine-2-carboxamide
N-methyl-1-[4-(4-methylphenoxy)piperidine-4-carbonyl]pyrrolidine-3-carboxamide
2-{imidazo[1,2-a]pyridin-2-yl}-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-chloro-N-ethyl-5-({[2-(ethylsulfanyl)ethyl]carbamoyl}amino)benzamide
6-ethyl-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-benzyl-1-(2-hydroxyethyl)-5-{[4-(propan-2-yloxy)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,5R)-6-(2,6-dimethoxypyridine-3-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-(azepan-1-yl)-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]butane-1,4-dione
2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
3-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-7-fluoro-1-(2-phenylethyl)-1,2-dihydroquinolin-2-one
{2-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]phenyl}methanol
1-(diethylamino)-3-[2-methoxy-4-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[2-(cyclohexylsulfanyl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-(4-methoxy-2-methylphenyl)-3-[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]propanamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
(3R,9aR)-8-(3,5-difluorobenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N,2-dimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)pyrido[2,3-d]pyrimidin-4-amine
(3-{2-[1-(dimethyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
(1S,5R)-3-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[1-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)-2-methylpropan-2-yl]morpholine
2-(3-fluoro-4-methoxyphenyl)-2-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetic acid
N-({7-[1-(4-chlorophenyl)cyclopropanecarbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(1H-imidazol-1-yl)acetamide
methyl 5-[(cyclohexylmethyl)amino]-3-acetamido-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-methyl-2-(5-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-1H-1,3-benzodiazole
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}({imidazo[1,2-a]pyridin-3-ylmethyl})methylamine
2-{1-cyclohexyl-5-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-5-yl]-1H-1,2,4-triazol-3-yl}acetamide
N-ethyl-2-[2-(2-phenylethyl)piperidin-1-yl]acetamide
1-{4-[(6-hydroxy-6-methylheptan-2-yl)amino]piperidin-1-yl}ethan-1-one