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8-methoxy-2-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}quinoline
4-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]urea
7-cyclobutaneamido-1-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-{2-[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}pyridine-3-carboxamide
methyl 3-[3-(2-chlorophenyl)propanoyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)piperidin-2-one
{3-[2-(1-cyclohexanecarbonylpiperidin-3-yl)-1H-imidazol-1-yl]propyl}dimethylamine
(4-benzyl-1-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)methanol
2-{[5-(1-ethyl-1H-pyrazol-5-yl)-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
8-{[3-(furan-2-yl)phenyl]methyl}-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)urea
9-methoxy-3-{[4-(propan-2-yloxy)phenyl]methyl}-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-methylacetamide
(2S,4R)-4-amino-N-(propan-2-yl)-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidine-2-carboxamide
N-[(4-chlorophenyl)methyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
[1-(2-methanesulfonylethyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
methyl 2-[1-(3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}phenyl)-N-methylformamido]acetate
N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
4-benzyl-3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
1-(naphthalen-1-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
4-{3-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
(2R,6R)-6-methyl-1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
4-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}thiomorpholine
3-methyl-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
ethyl 1-(3,5-dimethoxybenzoyl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
4-(4-ethyl-1H-pyrazol-5-yl)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
5-{[4-(3,4-dichlorophenyl)piperazin-1-yl]methyl}-2-(2-methoxyethyl)pyrimidine
(1R,2R)-2-[5-(2H-1,3-benzodioxol-5-yl)-3-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl]cyclohexan-1-ol
N-[(3S,4R)-1-(3-fluoro-4-methoxybenzenesulfonyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(oxolan-2-ylmethyl)benzamide
7-[2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)acetyl]-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-({7-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-[2-(methylamino)acetyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(4-{1-oxa-8-azaspiro[4.6]undecan-8-ylmethyl}thiophen-2-yl)ethan-1-one
N-[1-(3,5-dichlorophenyl)-2-hydroxyethyl]imidazo[1,2-a]pyridine-6-carboxamide
3-cyclopentyl-5-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazole
1-(2-cyclohexylethyl)-N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]furan-2-carboxamide
2-(4-chlorophenyl)-N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-{[3-({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}carbamoyl)phenyl]amino}acetic acid
1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-ol
2-(4-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)propanamide
3-(2-{2,7-diazaspiro[4.5]decan-7-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
[(3R,5R)-1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
N,1-dicyclopropyl-6-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
2-(2-methoxyphenyl)-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}acetamide
N,N-dimethyl-2-{[3-(4-methyl-1H-pyrazol-1-yl)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide