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1-[4-(cyclopropylmethyl)piperazin-1-yl]-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
1-{4-[3-(diphenylmethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperazin-1-yl}ethan-1-one
N-{2-methyl-1-[3-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-5-yl]propyl}acetamide
3-(1-benzyl-1H-imidazol-2-yl)-1-(1,3-thiazol-2-yl)piperidine
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(1H-indol-3-yl)propan-1-one
2-{2-[(furan-2-ylmethyl)sulfanyl]ethyl}-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-1-(2-methoxyethyl)-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
2-{1-[(2-ethoxyphenyl)methyl]-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
5-ethyl-N-[2-(2-fluorophenoxy)ethyl]-1,3,4-oxadiazol-2-amine
ethyl 5-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-[(2,6-difluorophenyl)methyl]-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R,4R)-3,4-dimethyl-1-[4-(4-methylpiperazin-1-yl)benzoyl]pyrrolidin-3-ol
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
3-(hydroxymethyl)-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidin-3-ol
1-[(3-chloro-4-ethoxyphenyl)methyl]-3-(methoxymethyl)piperidine
1-[(2-fluorophenyl)methyl]-N-{[4-(morpholin-4-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
[2-(2-fluoro-5-methoxyphenyl)phenyl]methanamine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3,6-dimethyl-1-benzofuran-2-carboxamide
[(3R,4S)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-(5-cyclopentaneamido-2-methylphenyl)-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide
N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]cyclohex-3-ene-1-carboxamide
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
(pyridin-3-ylmethyl)({[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl})(thiophen-3-ylmethyl)amine
2-[(4-methylpiperazin-1-yl)sulfonyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-6-(2,3-dihydro-1H-indene-5-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(2-chlorophenyl)ethyl]-2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]acetamide
[4-({1-[2-(pyrrolidin-1-yl)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
2-{3-[3-(morpholin-4-yl)-3-oxopropyl]piperidine-1-carbonyl}-4H-chromen-4-one
2-[5-(1H-1,2,3-benzotriazol-5-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-(propan-2-yl)pyridazin-3-amine
3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
N-benzyl-N-(3-hydroxy-2-methylpropyl)quinoline-8-carboxamide
N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(2-chloro-4-fluorophenoxymethyl)-N-(2-methoxyethyl)-N-methyl-1,3-oxazole-4-carboxamide
2-[(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-6-methoxyquinolin-2-yl)sulfanyl]acetic acid
2-[2-(dimethylamino)ethyl]-9-[2-(4-hydroxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-cyclohexyl-N-[1-(6-methoxynaphthalen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
2-methyl-5-(2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
N-{3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]phenyl}-3-(1,2-oxazolidin-2-yl)propanamide
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
3-methyl-6-{5-[(3,4,5-trimethoxyphenyl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
methyl 3-(2-methoxyacetamido)-5-{[1-(4-methoxyphenyl)propan-2-yl]amino}-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(2-fluorobenzoyl)-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(quinoline-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
(2S)-1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
5,7-dimethyl-N-{2-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-1-(4-methylpiperidin-1-yl)propan-1-one