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(2S,4R)-4-amino-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(3-{4-[(2-cyclohexylacetamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-2-methylfuran-3-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(pyridazine-4-carbonyl)piperidin-3-yl]propanamide
N-butyl-3-{[2-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-{4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-3-hydroxyphenyl}acetamide
9-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
4-[(3-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-4-methoxyphenyl)methyl]piperazin-2-one
4-(hydroxymethyl)-1-({4-[methyl(phenyl)amino]phenyl}methyl)azepan-4-ol
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(1-methyl-1,2,3,4-tetrahydroquinoline-6-carbonyl)piperidin-3-amine
N-cyclopropyl-5-methyl-1-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
3-(methylsulfanyl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
1-(3-chloro-5-fluorobenzoyl)-3-(2-ethylphenoxy)azetidine
6-amino-N-methyl-N-[4-(morpholin-4-yl)butyl]pyridine-3-carboxamide
N-cyclopentyl-6-fluoro-2-oxo-N-(thiophen-3-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[3-(1-methoxyethyl)phenyl]-N,N-dimethylpyrimidin-4-amine
6,6-dimethyl-1-(2-methylphenyl)-N-(oxan-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(1-{1-[2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
2-{4-[(dimethylamino)methyl]phenyl}-N,N,5-trimethylpyrimidin-4-amine
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]acetamide
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(4-ethylphenyl)methyl]-N-methylacetamide
N-(1H-1,2,3-benzotriazol-5-yl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]-3-(2-oxopyrrolidin-1-yl)propanamide
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
[1-(2H-1,3-benzodioxol-4-ylmethyl)-4-(oxan-2-ylmethyl)piperidin-4-yl]methanol
(1S,5R)-6-benzyl-3-[3-(pyridin-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4,6-dimethyl-1-(2-{4-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-1,2-dihydropyrimidin-2-one
1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
N-(1-{7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
6-oxo-1-(pyridin-2-ylmethyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidine-3-carboxamide
N-(2-chlorophenyl)-1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(thiophen-3-yl)ethan-1-one
2-(1H-1,3-benzodiazol-1-yl)-1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-{4-[(2-fluorophenyl)methyl]piperazin-1-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-[1-(2-methylbenzoyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide
6-(4-chlorophenyl)-N-(2,2,2-trifluoroethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl (2S)-1-[9-methoxy-7-oxo-3-(quinolin-7-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
N-[(3S)-2-oxoazepan-3-yl]-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)pyridine-2-carboxamide
methyl 2-{4-[5-(3-fluorobenzamido)-1H-pyrazol-1-yl]piperidine-1-carbonyl}benzoate
2-fluoro-N-{3-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-3-oxopropyl}benzamide
1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-3-(pyrrolidin-1-yl)piperidine
3-propyl-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-3-carboxylic acid
N-methyl-N-(3-phenylpropyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
methyl 3-(2-methoxypyridine-3-carbonyl)-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S,4R)-4-amino-N-methyl-1-{3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]propanoyl}pyrrolidine-2-carboxamide
N-(2-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
8-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
5-(3-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}propyl)-1H-1,2,3,4-tetrazole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-ol
3-butyl-1-methyl-4-(quinoxaline-6-carbonyl)piperazin-2-one