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N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
1-{2-[(1-methyl-3-phenyl-1H-pyrazol-5-yl)formamido]ethyl}piperidine-3-carboxamide
N-({1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
4-(6-methyl-1H-1,3-benzodiazol-2-yl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
4-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(piperidin-1-ylmethyl)-1,4-oxazepane
1-{4-[(1-methoxypropan-2-yl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
1-(3-{1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propyl)-1H-pyrazole
8-(2,2,2-trifluoroethanesulfonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide
4-(4-chlorophenyl)-1-[3-(pyridin-2-yl)azetidin-1-yl]butan-1-one
5-({2-[2-(furan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}methyl)-1-methylpyrrolidin-2-one
5-{4,6-dimethyl-11-oxo-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-13-yl}-2-methoxybenzoic acid
methyl 3-(2-fluorobenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(2-methoxyethyl)piperidin-1-yl]ethan-1-one
5-acetyl-N-[(2-ethoxyphenyl)methyl]-N-ethylthiophene-3-carboxamide
N-{2-[(2-chlorophenyl)formamido]ethyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]acetamide
1-(5-chloro-2-methoxyphenyl)-3-cyclopropyl-5-(pyrrolidine-1-carbonyl)-1H-1,2,4-triazole
5-chloro-1,3-dimethyl-4-{3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
2,3-difluoro-N-({8-[(4-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-[4-(2-phenylpropyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-amino-6-{4-[(dimethylamino)methyl]thiophen-2-yl}-4-(3-hydroxyphenyl)pyridine-3-carbonitrile
N-(2,2-dimethylpropyl)-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
1-(4-fluorophenyl)-4-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepane
1-(4-methylpiperazin-1-yl)-3-[1-(naphthalen-2-ylmethyl)piperidin-3-yl]propan-1-one
5-{[4-(4-methoxybutyl)piperazin-1-yl]methyl}-2-(3-methylphenyl)pyrimidine
N-{[3-(difluoromethoxy)phenyl]methyl}-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(1R,9S)-5-amino-3-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-[1-(propan-2-yl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-{[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-(3-fluorophenyl)acetamide
2-butyl-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-[3-(pyridin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-{2-[1-(3-chloro-1H-indole-2-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
8-(1-cyclopentylpiperidine-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-[(2-chlorophenyl)methyl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)spiro[2.3]hexane-1-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-methyl-1H-indole-2-carbonyl)piperidin-3-ol
8-[(2,3-dimethyl-1H-indol-7-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-4-(1H-pyrazol-4-yl)butanamide
3-cyano-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)benzamide
2-fluoro-N-({8-[2-(3-fluorophenyl)acetyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
2-(2H-1,3-benzodioxol-5-yl)-N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-hydroxy-1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
4-(dimethyl-1,3-oxazole-4-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(4-methoxyphenyl)methyl]-4-(4,4,4-trifluorobutanoyl)piperazin-2-one
4-[(2-hydroxybutyl)sulfamoyl]-N-(1H-imidazol-2-ylmethyl)benzamide
1-(4-{7-chloro-3-[(cycloheptylamino)methyl]quinolin-2-yl}piperazin-1-yl)ethan-1-one